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Title:
神経刺激性ステロイドの医薬組成物及びその使用
Document Type and Number:
Japanese Patent JP2008542419
Kind Code:
A
Abstract:
The present invention relates to a pharmaceutical composition, comprising 3±-hydroxy-3²-methoxymethyl-21-(1'-imidazolyl)-5a-pregnan-20-one or a pharmaceutically-acceptable salt or solvate thereof, and one or more pharmaceutically-acceptable excipients, wherein the composition provides steady state plasma levels of 3±-hydroxy-3²-methoxymethyl-21-(1'-imidazolyl)-5±-pregnan-20-one in a range of from 5 ng/mL to 500 ng/mL for a duration of from 6 h to 24 h following administration.

Inventors:
Woodward, Richard M.
Application Number:
JP2008515150A
Publication Date:
November 27, 2008
Filing Date:
June 09, 2006
Export Citation:
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Assignee:
Euro-Certique S.A.
International Classes:
A61K31/58; A61P25/18; A61P25/22; A61P25/24; A61P25/32; C07J43/00
Domestic Patent References:
JPS63122623A1988-05-26
JPS6330427A1988-02-09
JPH08183736A1996-07-16
Attorney, Agent or Firm:
Hiroshi Kobayashi
Eiji Katayama
Junko Kobayashi
Norio Omori
Yasuhito Suzuki