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Title:
一酸化窒素合成阻害剤として有用な2-アミノ-2-アルキル-5-ヘプテン酸及びヘプチン酸誘導体
Document Type and Number:
Japanese Patent JP2004509099
Kind Code:
A
Abstract:
The present invention relates to 2-amino-2-alkyl-5 heptenoic and heptynoic acid derivatives and their use in therapy, in particular their use as nitric oxide synthase inhibitors.

Inventors:
Hansen, Donald, Junior
Webber, Ronald Keith
Pizzel, Burnett S
James, Sickey
Mark A, Massa
Hagen, Timothy Jay
Grappler House, Margaret
Wang, Lijuane Jane
Berg Manis, Arija A.
Kramer, Stephen W.
Harinan, E Ann
Application Number:
JP2002526762A
Publication Date:
March 25, 2004
Filing Date:
September 15, 2001
Export Citation:
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Assignee:
Pharmacia Corporation
International Classes:
C07D265/32; A61K31/198; A61P1/02; A61P1/04; A61P1/16; A61P3/10; A61P9/00; A61P9/10; A61P11/00; A61P11/06; A61P17/02; A61P17/06; A61P19/00; A61P19/02; A61P19/08; A61P21/04; A61P25/04; A61P25/06; A61P25/28; A61P27/02; A61P27/06; A61P29/00; A61P35/00; A61P37/00; A61P43/00; C07C229/30; C07C237/16; C07C257/14; C07C259/14; C07C271/22; C07D271/06; C07D271/07; C07D413/06; C07F7/18; (IPC1-7): C07C257/14; A61K31/198; A61P1/02; A61P1/04; A61P1/16; A61P3/10; A61P9/00; A61P9/10; A61P11/00; A61P11/06; A61P17/02; A61P17/06; A61P19/00; A61P19/02; A61P19/08; A61P21/04; A61P25/04; A61P25/06; A61P25/28; A61P27/02; A61P27/06; A61P29/00; A61P35/00; A61P37/00; A61P43/00; C07C237/16; C07C259/14; C07C271/22; C07D265/32; C07D271/06; C07D413/06; C07F7/18
Domestic Patent References:
JP2000510820A2000-08-22
Foreign References:
WO1995025717A11995-09-28
Attorney, Agent or Firm:
Kazuo Shamoto
Tadashi Masui
Yasushi Kobayashi
Akio Chiba
Hiroyuki Tomita
Hiroko Ejiri