Title:
メシル酸イマチニブのＦ結晶形
Document Type and Number:
Japanese Patent JP5844508
Kind Code:
B2
Abstract:
The invention relates to the G-crystal form, I-crystal form and K-crystal form of the methanesulfonic acid addition salt of 4-(4-methylpiperazin-1-ylmethyl)-N-[4-methyl-3-(4-(pyridin-3-yl)pyrimidin-2-ylamino)phenyl]-benzamide, certain processes for their preparation, pharmaceutical compositions containing these crystal forms, their use in diagnostic methods or for the therapeutic treatment of warm-blooded animals, and their use as an intermediate or for the preparation of pharmaceutical preparations for use in diagnostic methods or for the therapeutic treatment of warm-blooded animals, especially humans.
Inventors:
Michael Muts
Application Number:
JP2008541641A
Publication Date:
January 20, 2016
Filing Date:
November 23, 2006
Export Citation:
Assignee:
Novartis Age
International Classes:
C07D401/04; A61K9/48; A61K31/506; A61K47/02; A61K47/04; A61K47/12; A61K47/32; A61K47/36; A61K47/42; A61P35/00; A61P35/02
Domestic Patent References:
| JP201474067A |
Foreign References:
| WO2005077933A1 | ||||
| WO2005095379A2 | ||||
| WO2004106326A1 | ||||
| WO1999003854A1 |
Other References:
岡野定舗編著,新・薬剤学総論(改訂第3版),南江堂,1987年4月10日,p.26,111,256,257
C.G.WERMUTH編,長瀬博監訳,最新 創薬化学 下巻,株式会社テクノミック,平成11年9月25日,p.452,453
C.G.WERMUTH編,長瀬博監訳,最新 創薬化学 下巻,株式会社テクノミック,平成11年9月25日,p.452,453
Attorney, Agent or Firm:
Hiroshi Kobayashi
Norio Omori
Kyoko Tamura
Yasuhito Suzuki
Norio Omori
Kyoko Tamura
Yasuhito Suzuki