Title:
AQUEOUS FORMULATION OF (2-HYDROXYMETHYL-INDANYL-4-OXY)-PHENYL-4, 4, 4-TRIFLUOROBUTANE-1-SULFONATE
Document Type and Number:
Japanese Patent JP2011098979
Kind Code:
A
Abstract:
To provide an aqueous formulation which includes (-)-(R)-3-(2-hydroxymethyl-indanyl-4-oxy)-phenyl-4, 4, 4-trifluorobutane-1-sulfonate and is suitable as an infusion solution or as a concentrate for producing the infusion solution.
The aqueous formulation includes (-)-(R)-3-(2-hydroxymethyl-indanyl-4-oxy)-phenyl-4, 4, 4-trifluorobutane-1-sulfonate (I) and cyclodextrin.
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Inventors:
KUEHN BERND
BRUECK ANTJE
KATAGAWA YOSHIFUMI
YASUI MASAMI
BRUECK ANTJE
KATAGAWA YOSHIFUMI
YASUI MASAMI
Application Number:
JP2011024007A
Publication Date:
May 19, 2011
Filing Date:
February 07, 2011
Export Citation:
Assignee:
BAYER SCHERING PHARMA AG
International Classes:
A61J1/10; A61K31/255; A61K9/00; A61K9/08; A61K9/10; A61K31/724; A61K47/02; A61K47/10; A61K47/12; A61K47/40; A61K47/48; A61P9/10
Domestic Patent References:
JP2001515470A | 2001-09-18 | |||
JP2000086539A | 2000-03-28 | |||
JPH11240833A | 1999-09-07 | |||
JPH07165616A | 1995-06-27 | |||
JPH05504783A | 1993-07-22 | |||
JP2005529864A | 2005-10-06 |
Other References:
JPN6009054921; Bela Szabo et al.: The Journal of Pharmacology and Experimental Therapeutics Vol. 297, No. 2, 2001, p. 819-826
Attorney, Agent or Firm:
Aoyama Aoi
Takuji Yamada
Michiko Matsutani
Mitsutaka Iwasaki
Yasushi Ochiai
Takuji Yamada
Michiko Matsutani
Mitsutaka Iwasaki
Yasushi Ochiai
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