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Title:
インテグリンアンタゴニストとしてのメタ−グアニジン、尿素、チオ尿素またはアザ環状アミノ安息香酸誘導体
Document Type and Number:
Japanese Patent JPH11510814
Kind Code:
A
Abstract:
The present invention relates to a class of compounds represented by the Formula Ior a pharmaceutically acceptable salt thereof, whereinA ispharmaceutical compositions thereof and methods of using such compounds and compositions as alphavbeta3 antagonists.

Inventors:
クレア,マイケル
コリンズ,ポール ダブリュ.
デサイ,ビピンチャンドラ エヌ.
ラッセル,マーク エイ.
リコ,ジョセフ ジー.
リンドマーク,リチャード ジェイ.
ルミンスキイ,ピーター,ジー
ロジャース,トマス イー.
Application Number:
JP51039797A
Publication Date:
September 21, 1999
Filing Date:
August 27, 1996
Export Citation:
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Assignee:
ジー.ディー.サール アンド カンパニー
International Classes:
A61K31/00; A61K31/155; A61K31/17; A61K31/195; A61K31/24; A61K31/335; A61K31/34; A61K31/341; A61K31/343; A61K31/357; A61K31/36; A61K31/38; A61K31/40; A61K31/403; A61K31/404; A61K31/4045; A61K31/41; A61K31/415; A61K31/4164; A61K31/4168; A61K31/4184; A61K31/4196; A61K31/44; A61K31/4406; A61K31/445; A61K31/4453; A61K31/4458; A61K31/47; A61K31/505; A61K31/513; A61K31/535; A61K31/5375; A61K31/54; A61K31/541; A61K31/70; A61K31/7028; A61K31/7034; A61K38/00; A61P5/38; A61P25/06; A61P35/00; A61P35/04; A61P43/00; C07C275/28; C07C275/42; C07C279/18; C07C279/24; C07C279/28; C07C311/19; C07C311/37; C07C313/34; C07C317/50; C07C323/59; C07C323/62; C07C323/63; C07C335/22; C07C335/28; C07D207/14; C07D207/22; C07D209/16; C07D211/72; C07D213/55; C07D213/61; C07D213/74; C07D215/14; C07D223/12; C07D231/06; C07D231/12; C07D231/14; C07D233/50; C07D233/64; C07D235/30; C07D239/14; C07D239/26; C07D239/54; C07D239/545; C07D249/14; C07D295/12; C07D295/14; C07D295/20; C07D295/215; C07D295/22; C07D307/54; C07D307/79; C07D307/81; C07D317/60; C07D317/64; C07D319/18; C07D319/20; C07D333/20; C07D333/24; C07D333/28; C07D401/12; C07D401/14; C07D405/10; C07D405/12; C07D413/12; C07D417/12; C07H15/203; C07K5/062; (IPC1-7): C07C275/42; A61K31/00; A61K31/195; A61K31/24; A61K31/335; A61K31/34; A61K31/36; A61K31/38; A61K31/40; A61K31/41; A61K31/415; A61K31/44; A61K31/445; A61K31/47; A61K31/505; A61K31/535; A61K31/54; A61K31/70; A61K38/00; C07C279/18; C07C279/24; C07C311/19; C07C313/34; C07C317/50; C07C323/59; C07C323/63; C07C335/22; C07C335/28; C07D207/22; C07D209/16; C07D211/72; C07D213/55; C07D213/61; C07D213/74; C07D215/14; C07D223/12; C07D231/12; C07D233/64; C07D235/30; C07D239/14; C07D239/26; C07D239/54; C07D249/14; C07D295/12; C07D295/14; C07D295/20; C07D295/22; C07D307/54; C07D307/79; C07D317/60; C07D317/64; C07D319/20; C07D333/20; C07D333/28; C07D401/12; C07D401/14; C07D405/12; C07D413/12; C07D417/12; C07H15/203; C07K5/062
Attorney, Agent or Firm:
浅村 皓 (外3名)