Title:
NOVEL DIAZABICYCLO [2.2.2]OCTANE DERIVATIVE
Document Type and Number:
Japanese Patent JP2018016544
Kind Code:
A
Abstract:
PROBLEM TO BE SOLVED: To provide a compound having an orexin receptor antagonistic effect, or a pharmaceutically acceptable salt thereof, or a solvate thereof, and a pharmaceutical composition containing the same as an active ingredient, and a pharmaceutical use thereof, particularly, a preventive and/or therapeutic agent for diseases associated with an orexin receptor, such as sleep disorders, psychiatric disorders, neurodegenerative diseases, memory disorders and eating disorders, in particular insomnia (insomniac condition), one of sleep disorders.SOLUTION: The present invention provides a compound represented by formula (I), or a pharmaceutically acceptable salt thereof, or a solvate thereof.SELECTED DRAWING: None
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Inventors:
HOTTA HIROMICHI
SAKURADA ISAO
SAKURADA ISAO
Application Number:
JP2014245240A
Publication Date:
February 01, 2018
Filing Date:
December 03, 2014
Export Citation:
Assignee:
MOCHIDA PHARM CO LTD
International Classes:
C07D471/08; A61K31/4995; A61K45/00; A61P25/20; A61P43/00
Attorney, Agent or Firm:
Koichi Tsujii
Sadao Kumakura
Atsushi Hakoda
Kenji Asai
Kazuo Yamazaki
Satsuki Ichikawa
Hironobu Hattori
Sadao Kumakura
Atsushi Hakoda
Kenji Asai
Kazuo Yamazaki
Satsuki Ichikawa
Hironobu Hattori