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Title:
置換オキソアザヘテロシクリル化合物
Document Type and Number:
Japanese Patent JP4829449
Kind Code:
B2
Abstract:
This invention is directed to oxoazaheterocyclyl compounds which inhibit Factor Xa, to oxoazaheterocyclyl compounds which inhibit both Factor Xa and Factor IIa, to pharmaceutical compositions comprising these compounds, to intermediates useful for preparing these compounds, to a method of directly inhibiting Factor Xa and to a method of simultaneously directly inhibiting Factor Xa and Factor IIa.

Inventors:
William Earl Ewing
Mikle Earl Becker
Yeon Me Choi-Sredeski
Heinz Double You Pauls
Way hay
Stephen M. Condon
Roderick S Davis
Barbara A. Honey
Alfredo Pspada
Christopher Jay Burns
John Zee
Iwen Lee
Mycle Earl Myers
One F Lau
Gregory Bee Poli
Application Number:
JP2001512520A
Publication Date:
December 07, 2011
Filing Date:
July 26, 2000
Export Citation:
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Assignee:
Aventis Pharmaceuticals Incorporated
International Classes:
A61K31/495; C07D241/08; A61K31/496; C07D401/14; A61K31/498; A61K31/502; A61K31/506; A61K31/517; A61K31/519; A61K31/5377; A61P7/02; A61P9/02; A61P9/04; A61P9/10; A61P19/02; A61P25/28; A61P35/00; A61P41/00; A61P43/00; C07D401/06; C07D403/06; C07D403/14; C07D405/14; C07D409/06; C07D409/12; C07D409/14; C07D413/14; C07D417/14; C07D471/04; C07D495/04
Domestic Patent References:
JP2000204081A2000-07-25
JPH08507072A1996-07-30
JPH11504651A1999-04-27
Attorney, Agent or Firm:
Junji Yuda
Chika Takagi
Kosuke Nishimura



 
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