Title:
2,6-DIOXO-3,6-DIHYDROPYRIMIDINE COMPOUND, AGRICULTURAL AND HORTICULTURAL BACTERICIDE, NEMATICIDE, AND MEDICAL AND VETERINARY ANTIFUNGAL AGENT
Document Type and Number:
WIPO Patent Application WO/2021/085389
Kind Code:
A1
Abstract:
The present invention addresses the problem of providing: a 2,6-dioxo-3,6-dihydropyrimidine compound which has excellent bactericidal activity, is safe, and can be industrially advantageously synthesized; and an agricultural and horticultural bactericide, nematicide, and medical and veterinary antifungal agent containing the same as an active ingredient. The compound according to the present invention is a compound represented by formula (II) or a salt thereof. In formula (II), each Y1 is an oxygen atom or a sulfur atom; Y2 is an oxygen atom or a sulfur atom; Z is a group represented by C-X1 or a nitrogen atom; X1 is a hydrogen atom, a halogeno group, or the like; X2 is a group represented by R1O-N=CR6- or the like; R1 is a substituted or unsubstituted linear C1-6 alkyl group or the like; R6 is a substituted or unsubstituted linear C1-6 alkyl group or the like; X3 is a substituted or unsubstituted linear C1-6 alkyl group, a substituted or unsubstituted linear C2-6 alkenyl group or the like; A is a substituted or unsubstituted C1-6 alkylene group, a substituted or unsubstituted C2-6 alkenylene group, or the like; and Q is a substituted or unsubstituted C6-10 aryl group or a substituted or unsubstituted 5-10 membered-ring heteroaryl group.
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Inventors:
TERANISHI TAKAAKI (JP)
KUWAHARA RAITO (JP)
MUNEI YOHEI (JP)
SHIMOMURA HAJIME (JP)
KAWASAKI TATSUHIRO (JP)
ISHIHARA TAKUMA (JP)
IWATA JUN (JP)
SAIGA TOMOYUKI (JP)
NISHINO CHIHIRO (JP)
KUWAHARA RAITO (JP)
MUNEI YOHEI (JP)
SHIMOMURA HAJIME (JP)
KAWASAKI TATSUHIRO (JP)
ISHIHARA TAKUMA (JP)
IWATA JUN (JP)
SAIGA TOMOYUKI (JP)
NISHINO CHIHIRO (JP)
Application Number:
PCT/JP2020/040135
Publication Date:
May 06, 2021
Filing Date:
October 26, 2020
Export Citation:
Assignee:
NIPPON SODA CO (JP)
International Classes:
C07D403/12; A01N43/54; A01N43/60; A01N43/647; A01N43/653; A01N43/707; A01N43/84; A01N55/10; A01P3/00; C07D239/54; C07D239/553; C07F7/10
Domestic Patent References:
| WO2013071169A1 | 2013-05-16 |
Foreign References:
| JPH09100269A | 1997-04-15 | |||
| US5859014A | 1999-01-12 | |||
| JP2010538068A | 2010-12-09 | |||
| JP2019195484A | 2019-11-14 | |||
| JP2020053191A | 2020-04-02 |
Other References:
ŞAHIN KADER, DURDAĞI SERDAR: "Identifying the Novel Pyrimidine-Based CDK2 Inhibitors as Anticancer Agents Using Text-Mining and Combined Molecular Modeling Approaches", JOURNAL OF THE TURKISH CHEMICAL SOCIETY SECTION A: CHEMISTRY, vol. 7, no. 2, 23 June 2020 (2020-06-23), pages 383 - 404, XP055822346, Retrieved from the Internet
See also references of EP 4053120A4
See also references of EP 4053120A4
Attorney, Agent or Firm:
HIROTA, Masanori (JP)
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