Title:
AROMATIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF
Document Type and Number:
WIPO Patent Application WO/2022/111513
Kind Code:
A1
Abstract:
Provided are an aromatic compound represented by formula A or a pharmaceutically acceptable salt thereof, and a preparation method therefor and the use thereof. The aromatic compound has a good inhibitory effect on KRAS, especially KRAS G12C.
Inventors:
XIANG JASON SHAOYUN (CN)
WANG SUYUE (CN)
LU ZHIJIAN (CN)
YANG SHUAI (CN)
FANG QI (CN)
HUANG TAO (CN)
YANG RUI (CN)
WANG SUYUE (CN)
LU ZHIJIAN (CN)
YANG SHUAI (CN)
FANG QI (CN)
HUANG TAO (CN)
YANG RUI (CN)
Application Number:
PCT/CN2021/132725
Publication Date:
June 02, 2022
Filing Date:
November 24, 2021
Export Citation:
Assignee:
HANGZHOU POLYMED BIOPHARMACEUTICALS INC (CN)
International Classes:
C07D401/04; A61K31/4709; A61K31/495; A61P35/00; C07D401/14; C07D413/04
Domestic Patent References:
WO2019213516A1 | 2019-11-07 | |||
WO2018217651A1 | 2018-11-29 | |||
WO2019051291A1 | 2019-03-14 |
Foreign References:
CN113061132A | 2021-07-02 | |||
CN111484477A | 2020-08-04 | |||
CN106488910A | 2017-03-08 |
Attorney, Agent or Firm:
SHANGHAI BESHINING LAW OFFICE (CN)
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