Title:
ENZYME INHIBITORS
Document Type and Number:
WIPO Patent Application WO1999046316
Kind Code:
A3
Abstract:
The present invention relates to compounds, compositions, and methods which are useful for the prevention and treatment of adverse health, skin, hair, and oral conditions. The compounds, compositions, and methods are also widely applicable for use in health, skin, hair, oral, beauty, and personal care applications. In particular, the present invention relates to compounds having structure (1): and the tautomers, acceptable salts, and biohydrolyzable amides, esters, and imides thereof, wherein A, Q, n, P, L1, L2, L3, L4, Z, X, B1 and B2 are defined herein.
Inventors:
MCIVER JOHN MCMILLAN
UNDERINER TODD LAURENCE
BATES TIMOTHY
UNDERINER TODD LAURENCE
BATES TIMOTHY
Application Number:
PCT/US1999/005314
Publication Date:
March 23, 2000
Filing Date:
March 11, 1999
Export Citation:
Assignee:
PROCTER & GAMBLE (US)
International Classes:
A61K8/00; A61K8/42; A61K8/49; A61K8/86; A61K31/155; A61K8/30; A61K31/167; A61K31/216; A61K31/505; A61K31/77; A61P3/04; A61P3/06; A61P3/10; A61P9/12; A61P43/00; A61Q17/00; C07C257/14; C07C257/18; C07C277/08; C07C279/18; C07D233/04; C07D239/06; C08G65/329; C08G65/48; A61K; C08G; C12N; (IPC1-7): C08G65/48; A61K31/155; C07C279/18; C07C257/18; C07C257/14; A61K31/77
Foreign References:
| EP0658585A2 | 1995-06-21 | |||
| US4556560A | 1985-12-03 |
Other References:
TAKERKART, GEORGES ET AL: "Preparation and properties of organophilic trypsin macroinhibitors. Diamidino-.alpha.,.omega.-diphenylcarbamylpolyethylene glycol", FEBS (FED. EUR. BIOCHEM. SOC.) LETT. (1974), 42(2), 214-17, XP000870353
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