Title:
FUSED RING DERIVATIVES USEFUL AS KRAS G12D INHIBITORS
Document Type and Number:
WIPO Patent Application WO/2022/188729
Kind Code:
A1
Abstract:
The disclosure relates to a KRAS G12D inhibitors of formula (I) or formula (IV), a composition containing the inhibitor and the use thereof.
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Inventors:
HAN HUIFENG (CN)
GAO PANLIANG (CN)
MA CUNBO (CN)
WANG PENG (CN)
LONG WEI (CN)
ZHANG HAO (CN)
ZHANG LEI (CN)
LIU DAN (CN)
GAO PANLIANG (CN)
MA CUNBO (CN)
WANG PENG (CN)
LONG WEI (CN)
ZHANG HAO (CN)
ZHANG LEI (CN)
LIU DAN (CN)
Application Number:
PCT/CN2022/079476
Publication Date:
September 15, 2022
Filing Date:
March 07, 2022
Export Citation:
Assignee:
JACOBIO PHARMACEUTICALS CO LTD (CN)
International Classes:
C07D498/16; A61K31/553; A61P35/00; C07D498/22
Domestic Patent References:
WO2021108683A1 | 2021-06-03 | |||
WO2021023154A1 | 2021-02-11 | |||
WO2021041671A1 | 2021-03-04 |
Foreign References:
CN110603258A | 2019-12-20 | |||
CN112074520A | 2020-12-11 | |||
CN112390818A | 2021-02-23 |
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