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Title:
PROCESS FOR PREPARATION OF MYCOPHENOLIC ACID AND ESTER DERIVATIVES THEREOF
Document Type and Number:
WIPO Patent Application WO2005105768
Kind Code:
A3
Abstract:
Provided are processes for preparation of mycophenolic acid.

Inventors:
KERI VILMOS (HU)
CZOVEK ZOLTAN (HU)
Application Number:
PCT/US2005/014347
Publication Date:
March 16, 2006
Filing Date:
April 26, 2005
Export Citation:
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Assignee:
TEVA GYOGYSZERGYAR RESZVENYTAR (HU)
TEVA PHARMA (US)
KERI VILMOS (HU)
CZOVEK ZOLTAN (HU)
International Classes:
C07D307/88; C07D307/00; C07D307/93
Domestic Patent References:
WO2001021607A22001-03-29
WO2004020426A12004-03-11
WO2001064931A12001-09-07
WO2002100855A12002-12-19
WO1997038689A21997-10-23
Foreign References:
GB1157099A1969-07-02
GB1158387A1969-07-16
US4452891A1984-06-05
EP0281713A11988-09-14
US5688529A1997-11-18
Other References:
SADHUKHAN A K ET AL: "OPTIMIZATION OF MYCOPHENOLIC ACID PRODUCTION IN SOLID STATE FERMENTATION USING RESPONSE SURFACE METHODOLOGY", JOURNAL OF INDUSTRIAL MICROBIOLOGY AND BIOTECHNOLOGY, BASINGSTOKE, GB, vol. 22, no. 1, January 1999 (1999-01-01), pages 33 - 38, XP000956451, ISSN: 1367-5435
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