Title:
SUBSTITUTED 1, 2, 4- TRIAZOLE DERIVATIVES AS OXYTOCIN ANTAGONISTS
Document Type and Number:
WIPO Patent Application WO2005082866
Kind Code:
A3
Abstract:
The present invention relates to a class of substituted triazoles of formula (I) with activity as oxytocin antagonists, uses thereof, processes for the preparation thereof and compositions containing said inhibitors. These inhibitors have utility in a variety of therapeutic areas including sexual dysfunction, particularly premature ejaculation (P.E.).
Inventors:
BROWN ALAN DANIEL (GB)
CALABRESE ANDREW ANTHONY (GB)
ELLIS DAVID (GB)
SMITH CHRISTOPHER RONALD (US)
CALABRESE ANDREW ANTHONY (GB)
ELLIS DAVID (GB)
SMITH CHRISTOPHER RONALD (US)
Application Number:
PCT/IB2005/000313
Publication Date:
April 13, 2006
Filing Date:
February 07, 2005
Export Citation:
Assignee:
PFIZER LTD (GB)
PFIZER (US)
BROWN ALAN DANIEL (GB)
CALABRESE ANDREW ANTHONY (GB)
ELLIS DAVID (GB)
SMITH CHRISTOPHER RONALD (US)
PFIZER (US)
BROWN ALAN DANIEL (GB)
CALABRESE ANDREW ANTHONY (GB)
ELLIS DAVID (GB)
SMITH CHRISTOPHER RONALD (US)
International Classes:
C07D249/08; C07D401/04; C07D401/06; C07D401/14; C07D403/06; C07D403/12; C07D405/04; C07D405/12; C07D405/14; (IPC1-7): C07D249/08; A61K31/4196; A61K31/4427; A61K31/4439; A61K31/444; A61K31/496; A61P5/10; C07D401/04; C07D401/14; C07D403/12; C07D405/04
Domestic Patent References:
| WO2001058880A1 | 2001-08-16 | |||
| WO2003053437A1 | 2003-07-03 |
Foreign References:
| JP2000063363A | 2000-02-29 |
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