PROCESS FOR MAKING BENZOXAZEPIN COMPOUNDS

Title:

PROCESS FOR MAKING BENZOXAZEPIN COMPOUNDS

Document Type and Number:

Japanese Patent JP2020114814

Kind Code:

A

Abstract:

To provide a novel process for making PI3K inhibitor compound GDC-0032.SOLUTION: There is provided a method for preparing PI3K inhibitor GDC-0032 having a structure described above and stereoisomers, geometrical isomers, tautomers and pharmaceutically acceptable salts thereof as well as a useful intermediate for preparing GDC-0032.SELECTED DRAWING: None

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Inventors:

REMY ANGELAUD
DANIAL R BEAUDRY
DIANE E CARRERA
SUSHANT MALHOTRA
TRAVIS REMARCHUK
FREDERIC ST-JEAN

Application Number:

JP2020032846A

Publication Date:

July 30, 2020

Filing Date:

February 28, 2020

Export Citation:

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Assignee:

HOFFMANN LA ROCHE

International Classes:

C07D498/04; A61P3/10; A61P29/00; A61P35/00; A61P37/02; C07C257/18; C07D233/90; C07D249/08; C07D267/14; C07D403/04

Attorney, Agent or Firm:

Sonoda/Kobayashi Patent Business Corporation

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