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Title:
CRYSTAL FORM OF ALLICIN-CYCLODEXTRIN INCLUSION COMPLEX COCRYSTAL, PREPARATION METHOD THEREFOR AND USE THEREOF
Document Type and Number:
WIPO Patent Application WO/2024/027219
Kind Code:
A1
Abstract:
The present invention relates to a crystal form of an allicin-cyclodextrin inclusion complex cocrystal, a preparation method therefor and a use thereof. The cyclodextrin in the crystal form of the allicin-cyclodextrin inclusion complex cocrystal is α-cyclodextrin, β-cyclodextrin, or γ-cyclodextrin. The crystal form of the allicin-cyclodextrin inclusion complex cocrystal has good water solubility and stable properties, and is not easily degraded.

Inventors:
HUANG YONGZHUO (CN)
SHEN HUAN (CN)
LIU ERGANG (CN)
Application Number:
PCT/CN2023/090363
Publication Date:
February 08, 2024
Filing Date:
April 24, 2023
Export Citation:
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Assignee:
ZHONGSHAN INST FOR DRUG DISCOVERY SIMM CAS (CN)
International Classes:
A61K31/724; C08L5/16; A61K36/8962; A61K47/40; A61P31/04
Foreign References:
CN107789345A2018-03-13
CN107802842A2018-03-16
CN101816744A2010-09-01
CN1565430A2005-01-19
US20160051594A12016-02-25
Attorney, Agent or Firm:
JIAQUAN IP LAW (CN)
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