| Document |
Document Title |
|
WO/1993/018006A1 |
The compounds of general formula (1) wherein R?1¿, R?2¿, R?3¿ are optionally substituted carbonyl and amide derivatives which are useful as inhibitors of retroviral proteases, and are effective in treating conditions characterized by ...
|
|
WO/1993/018093A1 |
New compounds have formula (I), in which one of the groups R?1¿ and R?2¿ is a nitro group, whereas the other is hydrogen, an alkyl group with 1 to 4 atoms or an alkoxy group with 1 to 4 atoms, R?3¿ and R?4¿ represent independently fr...
|
|
WO/1993/016986A1 |
Azo oxime ethers of general formula (I), in which X is CH or N, R1 is hydrogen, C1-C3alkyl, trifluoromethyl or cylclopropyl and R2 is aryl or heteroaryl, have an activity against phytopathogenic fungi. They can be used in the form of for...
|
|
WO/1993/015046A1 |
Carbamate having the formula (I), its plant-compatible acid addition and basic addition products, and fungicides containing the same are disclosed.
|
|
WO/1993/015090A1 |
Described are racemic optically active phosphorus compounds of formula (I), in which R is a hydroxy or protected hydroxy group, R1 is a hydroxy or protected hydroxy group or a lower alkoxy group and R2 is a lower alkyl, cycloalkyl or ary...
|
|
WO/1993/015091A1 |
Described are racemic optically active phosphorus compounds of the formula (I), in which R is a lower alkyl or lower alkoxy group and R1 is a lower alkyl, cycloalkyl or substituted phenyl group. The compounds of the formula (I) act, in t...
|
|
WO/1993/012072A1 |
The reaction time and ease of handling of reactants in the known process of forming optically active S-cyanohydrins by reacting aldehydes with hydrocyanic acid in the presence of the enzyme S-oxynitrilase and a solvent may be significant...
|
|
WO/1993/011117A1 |
Novel N-[2-(cyclic alkyl)phenyl]pyrazole-4-carboxamides useful as fungicides, methods of using said compounds, and fungicidal compositions containing them.
|
|
WO/1993/010094A1 |
A compound of the formula Het-NR-SO2-Ph2-A-Ph1 (COOH)(OH) and tautomic form, salts, solvates, C1-6 alkyl esters and pharmaceutical compositions of the compound. Ph1 and Ph2 are benzene rings with the proviso that carboxy and hydroxy are ...
|
|
WO/1993/010098A1 |
A process is disclosed for preparing methylpyrazoles from diacetylene and hydrazines. Diacetylene is separated by absorption from cracked gas, then reacted with hydrazines.
|
|
WO/1993/009095A1 |
Compounds of formula (I), wherein A represents C=C, S or O; Q represents a 5- or 6-membered unsaturated heterocycling ring having a nitrogen atom in the position adjacent to the point of attachment, 0-3 further heteroatoms selected from ...
|
|
WO/1993/009097A1 |
Constitution: a novel compound represented by general formula (1), wherein R1 represents -OR3 (R3 being H or alkyl), -NR4R5 (R4 and R5 being each H, alkyl or alkoxy), -NHCH(R6)COR7 (R6 being H or alkyl, and R7 being alkyl), -NHCH(R6)COOR...
|
|
WO/1993/009173A1 |
Use of 3-amino-2(benzoylamino)acrylic acid esters (I) in which R?1¿ is C¿1? to C¿20?-alkyl which may be interrupted by one or more non-adjacent O atoms or NR?5¿ groups and may bear one or more hydroxyl groups, C¿2? to C¿20?-alkenyl...
|
|
WO/1993/009098A1 |
Novel 4-cinnolinones of general formula (I) in which: A denotes oxygen or an NR3 grouping; R1 denotes: hydrogen, a C1-4 alkyl radical, a C1-4 phenyl alkyl radical or an aminoalkyl grouping; R2 is: a C2-5 alkyl, C3-5 alkenyl, C2-5 hydroxy...
|
|
WO/1993/007146A1 |
Benzo or pyridopyridazinones and pyridazinthiones of formula (I) wherein: X and Y are nitrogen or carbon, provided that at least one is carbon, and Z is oxygen or sulfur; R1 is hydrogen, lower alkyl, aryl, heteroaryl, or heterocycle lowe...
|
|
WO/1993/007116A1 |
Fungicidal compounds having formula (I), wherein W is CH3O.CH=CCO2CH3, CH3ON=CCONR3R4 or CH3ON=CCO2CH3 and stereoisomers thereof; n is 0 or 1; X is oxygen or sulphur; Z is oxygen, sulphur or NR1; R1 is hydrogen or alkyl optionally substi...
|
|
WO/1993/007109A1 |
Novel 3,4-dihydro-4-oxo-3-(prop-2-enyl)-1-phtalazineacetic acids and derivatives of formula (I) in which R1, R2 and R3 are the same or different and stand for H, a halogen or a linear or branched aliphatic, saturated or unsaturated radic...
|
|
WO/1993/004585A1 |
A herbicidal composition which comprises a phosphonate or phosphinate of formula (I), where R and R', which may be the same or different, each represent straight or branch-chained alkyl of 1 to 12 carbon atoms, and x and y are each 1 or ...
|
|
WO/1993/005021A1 |
A 4-amino(alkyl)cyclohexane-1-carboxamide compound represented by general formula (I), an isomer thereof, and a pharmaceutically acceptable acid addition salt thereof, wherein each symbol is as defined in the specification. These substan...
|
|
WO/1993/004043A1 |
Compounds of formula (I) wherein Ar, W, Z, Q, R1, U, and T are as set forth herein, are described. These compounds are active as agents against retroviruses and in particular against HIV.
|
|
WO/1993/004035A1 |
Described are compounds of formula (I), in which A is a valency bond or a straight or branched alkyl chain with 1 to 5 C-atoms; X is an -NR-CO (amide) or -NR-CO-NR- (urea) group in which R is a hydrogen atom or a C¿1?-C¿4? alkyl group;...
|
|
WO/1993/003022A1 |
Treatment of Aids, inhibition of the replication of HIV and related viruses, and formulations using thiourea derivative compounds or salts thereof are disclosed. Also disclosed are novel thiourea compounds.
|
|
WO/1992/021648A1 |
The present invention relates to compounds of formula (I).
|
|
WO/1992/020682A1 |
Substituted anilides of formula (I), wherein Q is one of (Q-1), (Q-2) and (Q-3), and R?1� to R?5�, Y, Z and Z?1� are as defined in the text, arthropodicidal compositions containing such compounds; and a method for controlling arthr...
|
|
WO/1992/020641A1 |
An optically active compound derived from a novel trifluorolactic acid, useful as a component of a ferroelectric liquid crystal composition, and a liquid crystal composition. A compound represented by general formula (I), wherein R?1� ...
|
|
WO/1992/019602A1 |
Compounds of formula (I), in which R1, R2 and X have the meanings given in the specification, and their salts and N oxides are new agents for the treatment of bronchial conditions and dermatitis.
|
|
WO/1992/017468A1 |
A pyridine derivative represented by general formula (I), a process for producing the same, and a herbicide comprising the same. In formula (I) W represents oxygen, sulfur, NH or N-C(O)B wherein B represents hydrogen or alkoxy; and Z rep...
|
|
WO/1992/017446A2 |
Compounds having aldose reductase inhibitory activity of formula (I) wherein X CH2, CH2CH2, -CHCH3, (a); Y=O or S; R1 is an optionally substituted phenyl, benzothiazol-2-yl, benzoxazol-2-yl, benzofuran-2-yl, benzothiophen-2-yl, thiazolop...
|
|
WO/1992/016510A1 |
The present invention relates to herbicidally, acaricidally and insecticidally active pyrazolidine-3,5-diones of formula (I), in which R1 is (a), (b) or (c); R2 and R3 independently of one another are C1-C6alkyl; C3-C6alkenyl; or C3-C6al...
|
|
WO/1992/015558A1 |
An indan derivative represented by general formula (1) or a pharmacologically acceptable salt thereof, wherein R1 represents C1 to C12 alkyl, benzyl, styryl, naphthyl, optionally substituted phenyl or optionally substituted thienyl; R2 r...
|
|
WO/1992/015307A1 |
Compounds of formula (I) wherein X and R1 have the meanings described in the specification, useful as antitumor agents.
|
|
WO/1992/013830A1 |
Fungicidal compounds having formula (I) and stereoisomers thereof, wherein A is hydrogen, halo, hydroxy, C1-4 alkyl, C1-4 alkoxy, C1-4 haloalkyl, C1-4 haloalkoxy, C1-4 alkylcarbonyl, C1-4 alkoxycarbonyl, phenoxy, nitro or cyano; R1 and R...
|
|
WO/1992/012136A1 |
A process for producing a hexahydropyridazine-1,2-dicarboxylic acid derivative represented by general formula (3) industrially in a good yield; wherein R represents alkoxy or aryl, which comprises reacting a hydrazinedicarboxylic acid de...
|
|
WO/1992/012137A1 |
The invention relates to novel, racemic and optically active 3(2H)-pyridazinone derivatives of general formula (I), wherein R1 means hydrogen; a C1-4alkyl group optionally substituted by an R5R6N- group where R5 and R6, being the same or...
|
|
WO/1992/012133A2 |
Compounds of formula (I), wherein Q, X, R?1�, R?2�, R?9� and Z are as defined in the text, including compositions containing said compounds and a method for using them to control arthropods.
|
|
WO/1992/012135A1 |
Optically substantially pure (-) enantiomer of [[4-(1,4,5,6-tetrahydro-4-methyl-6-oxo-3-pyridazinyl)phenyl]
hydrazono]propanedinitrile or pharmaceutically acceptable salt thereof, intermediates and a process for the preparation are descr...
|
|
WO/1992/010483A1 |
1-phenyl 1,4-dihydro 3-arylalkylamino 4-oxo pyridazines having geeral formula (I). Pharmaceutical compositions containing at least one of the compounds of general formula (I) as the active principle are also provided.
|
|
WO/1992/009578A1 |
This invention relates to substituted fused heterocyclic compounds of formula (I), which have utility as herbicides.
|
|
WO/1992/006963A1 |
Disclosed are new compounds of general formula (I), in which one of the substituents R1 and R2 is a methoxy, difluoromethoxy or ethoxy group and the other is a C4-C7 cycloalkoxy or C3-C7 cycloalkylmethoxy group, as well as the salts form...
|
|
WO/1992/004315A1 |
Monocyclic aryl compounds having selective LTB4 antagonists properties and comprising an amido substituent, a substituent group having a terminal carboxylic acid or derivative thereof and a lipophilic substituent, therapeutic composition...
|
|
WO/1992/002513A1 |
Heterocyclic compounds of formula (I), wherein R?1¿ and R?2¿ are each lower alkoxy, R?3¿ is substituted amino, etc., Y is CH or N and Z is CH or N, and pharmaceutically acceptable salts thereof which are useful as a medicament.
|
|
WO/1992/001765A1 |
The subject application discloses a chiral nonracemic composition of the general formula: R1-Ar-O-CH2-C*HX-C*HY-CH2-O-R2, wherein R1 is a tail group of two to sixteen carbons; Ar is an achiral FLC core of at least two rings; * denotes a ...
|
|
WO/1992/000968A1 |
Novel oxamide derivatives are described which inhibit the production of TNF and are useful in the treatment of disease states mediated or exacerbated by TNF production. The compounds of the present invention are also useful as inhibitors...
|
|
WO/1991/017983A1 |
Arthropodicidal tetrahydropyridazines of Formulae (I) and (II), wherein Q, X, X?1�, Y and G are as defined in the text, compositions containing them and their use in the control of arthropods.
|
|
WO/1991/017982A1 |
A novel substance matristatin represented by general formula (I) and a matristatin producing microorganism belonging to the genus Actinomadura, wherein R1 represents hydrogen or hydroxyl, R2 represents hydrogen or methyl, and R3 represen...
|
|
WO/1991/016314A1 |
A compound of general formula (I) and optionally a pharmaceutically acceptable salt thereof if it can form any salt, a process for the production thereof, and a medicinal composition containing the same as the active ingredient. These co...
|
|
WO/1991/016310A1 |
Antimicrobial quinolone thiourea compounds of general formula (I), wherein (1) A1, A2, A3, R1, R3, R4, and R6 form any of a variety of quinolone and related heterocyclic structures similar to those known in the art to have antimicrobial ...
|
|
WO/1991/016305A1 |
Heteroarylethenediyl or heteroarylethenediyl aryl compounds wherein the heteroaryl group can be mono- or bicyclic heteroaryl and the aryl group can be mono- or bicyclic heteroaryl or bi- or tricyclic carbocyclic, said compound optionally...
|
|
WO/1991/015123A1 |
The present disclosure is directed to substituted cyclohexanedione compounds, the preparation of said compounds, compositions containing said compounds and the use of said compositions in the selective pre- and postemergent kill and cont...
|
|
WO/1991/012241A1 |
A hydrazine derivative of formula (I), wherein A represents an optionally substituted phenyl, naphthyl or heteroaromatic group containing one or two nitrogen atoms, and R1 represents hydrogen, optionally substituted alkyl, or optionally ...
|
