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Matches 401 - 450 out of 3,730

Document Document Title
WO/2017/129139A1
Provided in the present invention are a sulfamic acid ester as an indoleamine-2,3-dioxygenase inhibitor, a preparation method therefor and a use thereof. The structure of the inhibitor in the present invention is shown in general structu...  
WO/2017/124822A1
Provided is a method for preparing IDO inhibitor epacadostat. The whole reaction route is simple, easy to control and has high yield.  
WO/2017/110865A1
Oxadiazole compounds indicated by formula (I) and the use of said oxadiazole compounds in plant disease control. [In the formula, Z represents OC(=X)NR2R3, OC(=X)YR4, or the like, R1 represents a halogen atom, a C1-4 alkoxy group, or the...  
WO/2017/110861A1
Provided is a plant disease control agent that contains a compound indicated by formula (I). [In the formula, G represents a benzene ring, a thiophene ring, a furan ring, a pyrazole ring, an imidazole ring, an oxazole ring, an isoxazole ...  
WO/2017/110862A1
The oxadiazole compound represented in expression (1) exhibits an excellent effect in controlling plant disease. (In the expression, G represents a benzene ring, a thiophene ring, a furan ring, etc., R1 represents a C1-C6 alkyl group, a ...  
WO/2017/109044A1
Compounds of the formula (I); wherein the substituents are as defined in claim 1, useful as a pesticides, especially as fungicides.  
WO/2017/111152A1
Oxadiazole compounds shown by formula (1) [in the formula, G represents a substituted or unsubstituted thiophene ring, furan ring, imidazole ring, oxazole ring, isoxazole ring, thiazole ring, oxadiazole ring, thiadiazole ring, pyridine r...  
WO/2017/103219A1
Compounds of the formula (I) wherein the substituents are as defined in claim 1, useful as a pesticides, especially as fungicides.  
WO/2017/103223A1
Compounds of the formula (I) wherein the substituents are as defined in claim 1, useful as a pesticides, especially as fungicides.  
WO/2017/104782A1
In order to provide a method for manufacturing a compound (1) or a pharmaceutically acceptable salt thereof, whereby yield can be improved, cost can be reduced by using an easily obtained, inexpensive starting material and efficiently re...  
WO/2017/102275A1
The invention relates to a compound of formula (I), an N-oxide or an agriculturally suitable salt thereof, wherein the variables are as defined in the specification, and their use as herbicides.  
WO/2017/101884A1
Disclosed are an indolamine 2,3-dioxygenase inhibitor having the structure of formula (I) and a preparation method and use thereof. The indolamine 2,3-dioxygenase (IDO) inhibitor is a (Z)-N'-hydroxy-N-benzamidine derivative, has a very h...  
WO/2017/097732A1
The invention relates to a compound of formula (I) wherein R1 to R3 are defined as in the description and in the claims. The compound of formula (I) can be used as a medicament.  
WO/2017/097246A1
A polymer comprising a repeating unit, which may further comprise one or more repeating units. The present subject matter also relates to a formulation comprising the polymer, and a fullerene, second polymer, or small molecule. The prese...  
WO/2017/093019A1
Substituted oxadiazoles for combating phytopathogenic fungi The present invention relates to oxadiazoles of formula (I), or the N-oxides and/or their agriculturally useful salts and to their use for controlling phytopathogenic fungi, and...  
WO/2017/089389A1
The invention relates to a compound of formula (I) wherein R1 and R2 are defined as in the description and in the claims. The compound of formula (I) can be used in the treatment of Human African TRypanosomiasis.  
WO/2017/085100A1
Substituted oxadiazoles for combating phytopathogenic fungi. The present invention relates the use of the compounds of the formula I or the N-oxides, or the agriculturally acceptable salts thereof for combating phytopathogenic harmful fu...  
WO/2017/085098A1
The present invention relates the compounds of the formula I, or the N-oxides, or the agriculturally acceptable salts thereof and to their use for combating phytopathogenic harmful fungi, wherein the variables are defined as given in the...  
WO/2017/087364A1
Novel hydrogen isotope-enriched 1,2,4-oxadiazole benzoic acid compounds, methods of their use and pharmaceutical compositions thereof are disclosed. The methods include methods of treating or preventing a disease ameliorated by modulatio...  
WO/2017/081312A1
The present invention relates to novel oxadiazoles of the formula (I), or the N-oxides and/or their agriculturally useful salts and to their use for controlling phytopathogenic fungi, or to a method for combating phytopathogenic harmful ...  
WO/2017/081311A1
Substituted oxadiazoles for combating phytopathogenic fungi The present invention relates to novel oxadiazoles of the formula I, or the N-oxides and/or their agriculturally useful salts and to their use for controlling phytopathogenic fu...  
WO/2017/081310A1
The present invention relates to novel oxadiazoles of the formula (I), or the N-oxides and/or their agriculturally useful salts and to their use for controlling phytopathogenic fungi, or to a method for combating phytopathogenic harmful ...  
WO/2017/080912A1
A thermodynamically stable crystal modification of 2-methyl-N-(5-methyl-1,3,4-oxadiazole-2-yl)-3-(methylsulfony l)-4-(trifluoromethyl)benzamide is described. Said thermodynamically stable crystal modification has particular advantages re...  
WO/2017/081309A1
Substituted oxadiazoles for combating phytopathogenic fungi The present invention relates to oxadiazoles of the formula I, or the N-oxides and/or their agriculturally useful salts and to their use for controlling phytopathogenic fungi, a...  
WO/2017/076739A1
The present invention relates to novel oxadiazoles of the formula I, or the N-oxides and/or their agriculturally useful salts and to their use for controlling phytopathogenic fungi, or to a method for combating phytopathogenic harmful fu...  
WO/2017/076742A1
The present invention relates to novel oxadiazoles of the formula I or an N-oxide and/or their agriculturally useful salts and to their use for controlling phytopathogenic fungi, or to a method for combating phytopathogenic harmful fungi...  
WO/2017/072247A1
Compounds of the formula (I) wherein the substituents are as defined in claim 1, useful as a pesticides, especially as fungicides.  
WO/2017/070084A1
The disclosed subject matter provides N- hydroxylsulfonamide derivative compounds of formulae (I), (II) or (III) as drawn below, pharmaceutical compositions comprising such compounds, kits comprising such compounds, and methods of using ...  
WO/2017/068136A1
The invention relates to 5,5'-bis(2,4,6-trinitrophenyl)-2,2'-bi(1,3,4-oxadiazole) and bis(2,4,6-trinitrobenzoyl)oxalohydrazide, an energetic active mass comprising or consisting of 5,5'-bis(2,4,6-trinitrophenyl)-2,2'-bi(1,3,4-oxadiazole)...  
WO/2017/065473A1
The present disclosure relates to novel compounds having histone deacetylase 6 (HDAC6) inhibitory activity, stereoisomers thereof or pharmaceutically acceptable salts thereof, the use thereof for the preparation of therapeutic medicament...  
WO/2017/055146A1
Described are acylated N-(1,2,5-oxadiazole-3-yl)-, N-(1,3,4-oxadiazole-2-yl)-, N-(tetrazole-5-yl)- and N-(triazole-5-yl)-aryl carboxamides of formula (I) and the use thereof as herbicides. In said formula (I), R, V, X, Y, and Z are group...  
WO/2017/059303A1
Provided herein are vinylogous thioester compounds and methods for using the compounds.  
WO/2017/055175A1
A method for synthesizing N-(1,3,4-oxadiazole-2-yl)aryl carboxamides of formula (I) is described, where the substituents represent groups such as hydrogen, alkyl, haloalkyl or aryl.  
WO/2017/055473A1
Compounds of the formula (I) wherein the substituents are as defined in claim 1, useful as a pesticides, especially fungicides.  
WO/2017/055469A1
Compounds of the formula (I) wherein, the substituents are as defined in claim 1, useful as a pesticides, especially as fungicides.  
WO/2017/050969A1
The present invention relates to modified fumarate molecules capable of activating HO-1 protein expression, their synthesis and their use in therapeutic applications, in particular their use in the treatment of inflammatory and cardiovas...  
WO/2017/049245A2
The disclosure features novel lipids and compositions involving the same. Nanoparticle compositions include a novel lipid as well as additional lipids such as phospholipids, structural lipids, and PEG lipids. Nanoparticle compositions fu...  
WO/2017/035662A1
Described herein is a genetic modifier of cystic fibrosis (CF), which may serve as a predictor of the efficacy of a CFTR-directed therapy. SNPs rs7512462 or rs2869027 in non-coding regions of SLC26A9 are shown to correlate with CF lung d...  
WO/2017/032728A1
The invention relates to substituted ketoxime benzoylamides of general formula (I) as herbicides. In said formula (I), R1', R2', X, Y and W represent groups such as hydrogen, organic groups such as alkyl, and other groups such as halogen...  
WO/2017/031325A1
The present disclosure relates to oxadiazine compounds, pharmaceutical compositions comprising an effective amount of an oxadiazine compound and methods for using an oxadiazine compound in the treatment of a neurodegenerative disease, co...  
WO/2017/018805A1
The present invention relates to novel compounds having histone deacetylase 6 (HDAC6) inhibitory activity, stereoisomers thereof or pharmaceutically acceptable salts thereof, the use thereof for the preparation of therapeutic medicaments...  
WO/2017/018803A1
The present invention relates to novel compounds represented by the formula I having histone deacetylase 6 (HDAC6) inhibitory activity, stereoisomers thereof or pharmaceutically acceptable salts thereof, the use thereof for the preparati...  
WO/2017/018804A1
The present invention relates to: a novel compound having a histone deacetylase 6 (HDAC6) inhibitory activity; an optical isomer thereof or a pharmaceutically acceptable salt thereof; a use thereof for preparing a therapeutic pharmaceuti...  
WO/2017/010399A1
Provided are compounds having RORγt inhibitory effects represented by formula (I). Compounds represented by formula (I) (wherein L represents -NR1ACO-, -SO2- or the like, A represents a substituted or unsubstituted aromatic carbocyclic ...  
WO/2017/005564A1
The invention relates to N-(1,3,4-oxadiazol-2-yl) aryl carboxamide derivatives of the general formula (I) as herbicides. In said formula (I), V, X, and Z represent groups such as hydrogen, and organic groups such as alkyl, and other grou...  
WO/2017/004964A1
The present invention provides a novel preparation method of a 3-[5-(2-Fluorophenyl)-1,2,4-oxadiazol-3-yl]benzoic acid as a drug for preventing muscular dystrophy and an intermediate compound. The preparation method has a reasonable prod...  
WO/2017/004608A1
The invention is directed to Compounds of Formula (I): wherein each variable is defined herein, as well as methods of making and using the compounds as agonists of S1P1 and/or S1P5 for instance for treating graft versus host disease and ...  
WO/2017/004610A1
Disclosed are tercyclic S1P3-sparing, S1P1 receptor agonists, as well as processes for making and methods of using the same. Poor solubility and cationic amphiphilic drug- likeness were liabilities identified for a lead series of S1P3-sp...  
WO/2016/198507A1
Compound of formula (I) wherein A is selected from (i), where RF1 is H or F; (ii); (iii) a N-containing C6 heteroaryl group; and B is (B), where X1 is either CRF2 or N, where RF2 is H or F; X2 is either CR3 or N, where R3 is selected fro...  
WO/2016/201168A1
The present disclosure relates to oxadiazine compounds, pharmaceutical compositions comprising an effective amount of an oxadiazine compound and methods for using an oxadiazine compound in the treatment of a neurodegenerative disease, co...  

Matches 401 - 450 out of 3,730