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JPH0656807A |
PURPOSE: To provide a new compd. which is effective to treat, prevent or control renin-associated hypertension, hyperaldosteronism, congestive heart failure and galucoma. CONSTITUTION: This compd., for example a compd. expressed by formu...
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JPH0648943A |
PURPOSE: To obtain a medicine containing as specified aryl-substd. rhodamine as an effective component for the treatment and prevention of I-type diabetes. CONSTITUTION: This medicine contains a compd. expressed by formula I or its medic...
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JPH068290B2 |
Fungicidally effective aminomethyl heterocyclic compounds of the formula in which X represents oxygen or sulphur, R represents hydrogen or alkyl, or represents in each case optionally substituted cyclohexyl or phenyl and R1 and R2 indepe...
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JPH06500994A |
Compounds of formula (I), wherein R<4> is hydrogen and either R<5> is hydrogen and R<6> is hydroxyl or R<5>, R<6> and the carbon to which they are attached together form a carbonyl group; or R<6> is hydrogen and R<4> and R<5> together fo...
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JPH069614A |
PURPOSE: To obtain substd. dibenz-oxa-thiocinone-12-oxides and -12,12-dioxides useful in the preparation of circulation-influencing medicaments. CONSTITUTION: The substd. dibenz-oxa-thiocinone-12-oxides and -12,12-dioxides are compds. of...
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JPH06500099A |
PCT No. PCT/US91/05028 Sec. 371 Date Dec. 7, 1992 Sec. 102(e) Date Dec. 7, 1992 PCT Filed Jul. 22, 1991.A class of heterocyclic amino-alcohol compounds is described for treatment of CNS-related diseases, namely, for use as a neuroprotect...
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JPH05507936A |
PCT No. PCT/FR91/00549 Sec. 371 Date Dec. 10, 1992 Sec. 102(e) Date Dec. 10, 1992 PCT Filed Jul. 8, 1991 PCT Pub. No. WO92/00975 PCT Pub. Date Jan. 23, 1992. (I) A method for preparing cyclic sulphates having general formula (I), wherein...
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JPH0580471B2 |
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JPH05294964A |
PURPOSE: To obtain the subject compds. useful for antiviral agents or the like in high yield by bringing a specified racemic compd. to react under specified conditions, thereafter eliminating a protecting group and efficiently attaining ...
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JPH05294958A |
PURPOSE: To provide a new compound useful as a mercury ion removing agent and a silver halide dissolving agent. CONSTITUTION: The compound of formula I (X is 0 or S; (n) is 1-5; R is phenyl or phenyl bonded to a polymer via a bivalent gr...
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JPH05271139A |
PURPOSE: To provide two new kinds of the subject compds. extremely adequate as starting raw materials for production of mixtures composed of carbocyclic nucleosides of natural and unnatural series or their racemates. CONSTITUTION: The co...
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JPH0567151B2 |
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JPH05247027A |
PURPOSE: To obtain 1,3-oxathiolane-2-thionederivative under mild reaction conditions in good yield. CONSTITUTION: The objective method for producing 1,3-oxathiolane-2-thione is characterized by reacting an epoxy compound with carbon disu...
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JPH05239013A |
PURPOSE: To produce a sulfoalkylating agent inexpensive and physiologically harmless. CONSTITUTION: The sulfoalkylating agent is derived from a hydroxyalkanesulfonic acid or a corresponding alkanesultone selected from a group consisting ...
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JPH0560830B2 |
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JPH05222005A |
PURPOSE: To provide the subject compound which has the ability to inhibit angiotensinogen-cleaving action of the natural proteolytic enzyme, renin and is useful for preventing and treating renin-associated hypertension, hyperaldosteronis...
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JPH0555507B2 |
This invention relates to novel imidazole and triazole substituted oxathiolane compounds and compositions containing said compounds having fungicidal and plant growth regulant activity and methods for preparing same. The compounds may be...
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JPH05194480A |
PURPOSE: To prepare a new heterocyclic compd. having insecticidal activity an acaricidal activity. CONSTITUTION: The compd. of formula I [R1 is H or a halogen; R2 is a halogen, R3 is H, a halogen or an alkyl; R4 and R5 are each H, an alk...
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JPH05186451A |
PURPOSE: To obtain a dye compd. capable of bonding the dye to a solid support without deteriorating the pH sensitivity of the dye and preventing the leaching of the dye when the support is utilized as the pH sensor of optical fibers. CON...
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JPH0544946B2 |
Cyclic disulfonic ester bifunctional cross-linking compounds effective in treating certain types of cancers are described. Initial nucleophilic reaction with the compound produces a negatively charged sulfonic acid end-group which remain...
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JPH0543704B2 |
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JPH05504139A |
PCT No. PCT/EP91/00075 Sec. 371 Date Jul. 20, 1992 Sec. 102(e) Date Jul. 20, 1992 PCT Filed Jan. 17, 1991 PCT Pub. No. WO91/10659 PCT Pub. Date Jul. 25, 1991.Oxathiane derivatives of formula (I) in which R represents alkyl and A represen...
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JPH05140063A |
PURPOSE: To provide the subject new compounds showing an inhibitory effect on depression of Ca-concentration or collagen fiber content in bone and useful as a medicine for preventing and improving bone-absorption diseases such as maligna...
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JPH05140131A |
PURPOSE: To obtain a new ferroelectric liquid crystalline compound, excellent in thermal stability, having great spontaneous polarization and most suitable for producing a liquid crystal device having a high speed of response and having ...
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JPH0535151B2 |
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JPH0514714B2 |
A benzoxathiin derivative having the formula wherein R<1> represents hydrogen atom or a lower alkyl group, and R<2> represents a lower alkyl group or an aralkyl group, or a pharmaceutically acceptable acid addition salt thereof Pharmaceu...
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JPH0543572A |
PURPOSE: To obtain the title compound useful as a sulfoalkylating agent for cyclic tertiary amines of spectral sensitizing coloring matter for photography and dye for photography and intermediates for medicine and surfactant by using bis...
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JPH0513153B2 |
Highly effective diuretic antihypertensives, i.e., benzofuran or benzothiophene derivatives having a substituted propenoyl group at the 5-position, which are classified into loop diuretics with less adverse effects and can be administere...
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JPH0512339B2 |
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JPH0511115B2 |
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JPH059170A |
PURPOSE: To obtain a new compound useful as an excellent antitumor agent. CONSTITUTION: A compound shown by formula I [X1 and X2 are O, S(O)n ((n) is 0-2), N(R3) (R3 is lower hydrocarbon) or methylene; Y 18 NH-C (=Z)-NH (Z is O or S), N=...
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JPH059187A |
PURPOSE: To provide the subject new compound useful as a dye precursor and giving a heat-sensitive recording material having excellent whiteness, storability and color-developing property. CONSTITUTION: The compound of formula I {R is 4-...
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JPH0481589B2 |
Compounds of formula (I):in which:R1 represents a hydrogen atom, an alkyl group, a substituted alkyl group, a C2-C6 alkenyl group, an aryl group, a substituted aryl group or a (C1-C6 alkoxycarbonyl group; R2 represents a hydrogen atom, a...
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JPH04342586A |
PURPOSE: To provide the subject novel compound as a herbicide. CONSTITUTION: A compound of formula I [R1 is halogen, (halogen-substituted) alkyl, alkoxy, etc.; R2, R3 are H, alkyl; R4 is alkyl; X1, X2 are O, S; Y1, Y2 are methyl, methoxy...
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JPH0465826B2 |
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JPH0462315B2 |
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JPH0462314B2 |
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JPH0458476B2 |
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JPH04244079A |
PURPOSE: To obtain a new compound having agrochemical activity as insecticide and miticide. CONSTITUTION: This compound of the formula I, e.g. 2,6-difluoro-N[[[2-(2- fluorophenyl)-1,3-benzodioxan-6-yl]amino] carbonyl[benzamide is obtaine...
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JPH04243853A |
PURPOSE: To produce a new 4-aminobutyric acid compound which can be used to treat spasmodic diseases and old age related diseases. CONSTITUTION: The new compound is the compound of formula I (wherein R1 is OH, NH2, lower alkylamino, lowe...
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JPH04504568A |
The present invention provides a process for the conversion of a reactant into a reaction product in the presence of a solid acid catalyst comprising one or more fluorine atoms, sulfo radicals and phosphono radicals, each such radical be...
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JPH04217961A |
PURPOSE: To provide new compounds which inhibit the angiotensinogen-cutting action of the natural proteolytic enzyme, renin. CONSTITUTION: This compound is represented by formula I [A is H, Het (Het is 5-7 membered monocyclic ring having...
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JPH0448222B2 |
PURPOSE:To attain high sensitivity and to improve the characteristics after repeated used by forming a photosensitive layer contg. a specified salt com pound. CONSTITUTION:A photosensitive layer contg. a thulium salt compound represented...
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JPH0448220B2 |
PURPOSE:To obtain an org. semiconductor film having high sensitivity by contg. oxathiillium salt compd. CONSTITUTION:A titled body is constituted with an electrophotographic sensitive body provided with the photoconductive film contg. th...
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JPH04503073A |
Oligopeptide compounds or oligopeptide analogue compounds of the formula A-B-D-E-G-J-L-M-Q-T are ligands for the anaphylatoxin receptor and are useful in the treatment of inflammatory disease states. Also disclosed are anaphylatoxin rece...
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JPH04124179A |
PURPOSE: To simply obtain in high yield the title compound in high concentration by reaction of each specific two kinds of compound in the presence of a base followed by reaction of the resulting product with another specific compound. C...
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JPH0417957B2 |
A compound of the formula:(wherein Az is imidazolyl or triazolyl;R is C1-C5 Alkyl or phenyl optionally substituted by 1 to 3 members selected from halogen, C1-C5 alkyl, and C1-C5 alkoxy;X1 and X2 each is hydrogen, halogen, C1-C5 alkyl, o...
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JPH045672B2 |
Novel 1,5-benzoxathiepin derivatives of the formula: [wherein R1 and R2 are independently hydrogen, halogen, hydroxy, lower alkyl or lower alkoxy; R3 and R4 are independently hydrogen, optionally substituted lower alkyl or optionally sub...
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JPH045673B2 |
Novel 1,5-benzoxathiepin derivatives of the formula: [wherein R1 and R2 are independently hydrogen, halogen, hydroxy, lower alkyl or lower alkoxy; R3 and R4 are independently hydrogen, optionally substituted lower alkyl or optionally sub...
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JPH0429987A |
PURPOSE: To obtain the subject compound useful as drugs, etc., antioxidants, etc., in high yield and purity using simple operation by reacting an aldehyde with a specific alcohol in the presence of an amine.hydrochloride used as a cataly...
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