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JP4371054B2 |
A novel production method of quinolinecarbaldehydes (IV), which includes reacting aminobenzophenones (I) with beta -ketoaldehyde derivative (II) in the presence of an acid to give quinolinecarbaldehyde derivative (III), and then hydrolyz...
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JP4373622B2 |
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JP2009532437A |
The present invention relates to N-cyclopropyl-sulfonylamide derivatives of formula (I) wherein the substituents are cyclic groups, their process of preparation, their use as fungicide active agents, particularly in the form of fungicide...
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JP4316497B2 |
This invention relates to organic catalysts comprising iminium or oxaziridinium moieties, cleaning compositions comprising such catalysts; and processes for making and using such catalysts and cleaning products.
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JP4280276B2 |
The present invention provides enantiomerically pure ²-D-(-)-dioxolane-nucleosides. The enantiomerically pure dioxolane nucleosides are active HIV agents, that are significantly more effective than the prior prepared racemic mixtures of...
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JP4282261B2 |
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JP4281030B2 |
To provide a lithium secondary battery with high safety and high reliability. Aluminum or an aluminum alloy is used as a positive current collector, and an electrolyte or a polymer gel electrolyte contains at least one of compounds repre...
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JP4278345B2 |
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JPWO2007049798A1 |
Equation (I)[In the formula, Ar indicates a benzene ring, etc., and X1Indicates nitrogen atom, sulfur atom, etc., and R1Indicates an aryl group, etc., and X2Is equation (II)(In the formula, R4And R5Indicates a lower alkyl group, etc., m ...
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JP4249393B2 |
Processes for the preparation of 1,3-oxathiolane nucleosides are provided that include efficient methods for the preparation of the 1,3-oxathiolane ring and subsequent condensation of the 1,3-oxathiolane with a pyrimidine or purine base....
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JP4240531B2 |
Heterocyclic substituted benzoyl derivatives of the formula where Z is a 5-membered or 6-membered heterocyclic, saturated or unsaturated radical containing one to three hetero atoms selected from the group consisting of oxygen, sulfur an...
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JP2009046478A |
To provide a compound exhibiting excellent controlling effects against noxious arthropods.The imidate compound represented by formula (I) [wherein Z is an optionally substituted carbocyclic group having 3-14 ring-constituting atoms, or t...
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JP2009040788A |
To provide a synthesizing method for an HIV-protease inhibitor, nelfinavir mesylate and a new intermediate for synthesizing it.The synthesizing method uses a new intermediate such as a compound 7a.
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JP4226842B2 |
A high resolution resist material comprising an acid generator is provided so that high sensitivity and high resolution for high energy rays of 300 nm or less, small line-edge roughness, and excellence in heat stability and storage stabi...
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JP4215986B2 |
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JP4212576B2 |
To provide a 3-oxa-2-thiatricyclo[4.2.1.04,8]nonane derivative. The nonane derivative represented by formula [Rais H or an alkyl; R1, R2, R3, R4are each H, an alkyl; R5, R6, R7are H, an alkyl, a substituted oxycarbonyl, cyano; X is methy...
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JP2008308494A |
To provide a new compound having a COMT (catechol-O-methyl transferase)-inhibiting action.Provided are the compound represented by general formula (I) [wherein, R1 and R2 are each H, a lower acyl, a lower alkoxycarbonyl, or the like; R3 ...
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JP4195074B2 |
[Object] To provide a substituted cycloalkene derivative having an action to supress intracellular signal transduction or cell activation induced by endotoxin and to suppress cell responses due to the intracellular signal transduction an...
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JP2008260760A |
To provide a pharmaceutical composition excellent in prevention and/or therapy of diseases such as septicemia, a compound able to be used for the same and a method for producing the same.The pharmaceutical composition contains a compound...
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JP4170631B2 |
The present invention relates to the perfumery and flavor industry. It concerns more particularly the use of a compound of formula (I) as perfuming or flavoring ingredient wherein R<1> and R<2> represent simultaneously or a independently...
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JP2008538210A |
Compounds of the formula (I) in which the substituents are as defined in claim 1 are suitable for use as microbiocides.
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JP4153031B2 |
The invention relates to compounds of the formulae:processes for their preparation, polymers, co-polymers or block co-polymers containing them or their use as monomers or co-monomers in free radical polymerisation and in the manufacture ...
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JP4129993B2 |
Novel compounds are provided which are inhibitors of MTP and thus are useful for lowering serum lipids and treating atherosclerosis and related diseases, and have the structure (I) or (IA) or (IB) including pharmaceutically acceptable sa...
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JP4125418B2 |
Benzodioxin and benzoxathiin derivatives of formula (I), their enantiomers, diastereoisomers, and salts with acids and bases are new: X, Y = S, O, CHq, CHSO or SO2, such that X, Y may not both be CHq; q = 0-2; Z = O or CH2; n = 0-4; A = ...
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JP4111638B2 |
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JP2008521850A |
Compounds of the formula wherein the substituents are as defined in the claims, are useful as fungicides.
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JP4108851B2 |
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JP4108645B2 |
The present invention relates to a method of preparing BCH-189 and various analogues of BCH-189 from inexpensive precursors with the option of introducing functionality as needed. This synthetic route allows the stereoselective preparati...
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JP2008519824A |
Compounds of formula 1: are disclosed, wherein V is CH2; W is S(O)m; m is the integer 0, 1 or 2; U is O, C(O), CR13R14 or NR15; where R13 is H, alkyl; R14 is H, OH, OR13 or OCOR13; R15 is H, alkyl, cycloalkyl, alkenyl, C(O)R13, C(O)OR13 ...
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JP2008518910A |
Novel opiate intermediate compositions and methods of synthesis that include changing the substitution pattern on the aromatic ring of the pre-Grewe intermediate are provided. The intermediates are morphinane derivatives of formula (10),...
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JP2008512438A |
This invention is directed to compounds of formula Ia, Ib or Ic and to pharmaceutical compositions thereof:
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JP4079929B2 |
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JP4056558B2 |
The invention relates to a diastereoselective process for the preparation of compounds of formula (1), wherein W is S, S=O, SO2 or O; X is S, S=O, SO2 or O; R1 is hydrogen or acyl, and R2 is a purine or pyrimidine base or an analogue or ...
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JP2007326863A |
To provide a compound useful as a retroviral protease inhibitor, and in particular as an inhibitor of HIV protease; and to provide a method for treating retroviral infection by the compound. The compound is represented by the chemical fo...
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JP4015997B2 |
A purification method is disclosed for a predetermined water-insoluble extractant present in a liquid phase composition that additionally contains one or more additional extractants, synthesis reaction starting materials, and reaction by...
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JP2007530657A |
Materials and methods for preparing P-chirogenic monophospholanes and bisphospholanes are disclosed. The methods employ stereoselective cyclization to generate the phospholane rings followed by pyramidal inversion to access a variety of ...
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JPWO2005080322A1 |
The present invention relates to a novel fluorene derivative or a salt thereof, which is characterized by a structure in which a functional group such as a guanidino group is bonded to a fluorene skeleton via a carbonyl group. The compou...
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JP3995292B2 |
To obtain a new compound useful as a material for silver-halide photosensitive materials. This sultone compound of formula I (La1 is methylene; Lb1 and Lc1 is each methine; k1 is 2 or 3 provided that Lb1 and LC1 are unsubstituted methine...
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JP3989554B2 |
The invention relates to a group of new piperazine and piperidine compounds having interesting pharmacological properties. It has been found that compounds of formula (a) wherein A represents a heterocyclic group of 5-7 ring atoms wherei...
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JP3982879B2 |
A substituted carboxanilide derivative provided by the invention and represented by the formula (1): wherein A is is a hydrogen atom or methyl, B is a methyl or ethyl, and Het is 1-methyl-3-substituted-4-pyrazolyl or 2-methyl-4-substitut...
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JP2007217425A |
To provide a method for the diastereoselective synthesis of nucleoside analogs. The invention provides a method for the stereoselective production of a compound of formula (I) (W is S, S=O, SO2or O; X is S, S=O, SO2or O; R1is hydrogen or...
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JP2007210924A |
To provide a bactericidal composition by overcoming problems such that conventionally provided bactericidal compositions have several problematic points on practical usage such as either any of preventive effect and treating effect is in...
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JP2007521255A |
The present invention is based, at least in part on the discovery of therapeutic agents capable of preventing, inhibiting or modulating abnormal processing, misfolding or aggregation of protein. The therapeutic agents of the invention ma...
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JP2007520505A |
The invention relates to novel carboxamides of formula (I), in which M represents a phenyl ring, pyridine ring or pyrimidine, pyridazine or pyrazine ring, respectively monosubstituted by R8, or represents a thiazole ring substituted by R...
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JP2007520500A |
New haloalkyl carboxamides of formula (I) in which R, R1, R2, R3, R4, M and A have the meanings specified in the description, several processes for synthesizing these materials and their use in combating undesirable microorganisms, as we...
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JP3922656B2 |
To obtain a new compound useful as a material for silverhalide photosensitive materials. This sultone compound of formula I (A1 and A2 are each H, an alkyl, aryl, heterocyclic ring provided that either of Al1 and A2 is not H; La is methy...
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JP2007508337A |
This invention is related to compounds of general formula I wherein X is oxygen or sulphur or a NR<7> group; R<1> is C3-C8 alkyl, or C1-C8 alkyl substituted by phenoxy or phenyl, both phenoxy or phenyl being optionally substituted by o...
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JP2007505950A |
The invention provides novel non-beta-lactam inhibitors of beta-lactamases. In particular, the invention provides boronic acid-based compounds set forth in the specification. These compounds may be used with beta-lactam antibiotics to ba...
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JP3892912B2 |
PURPOSE: To obtain a method for measuring a substance to be inspected in a medium suspected of containing the substance to be inspected. CONSTITUTION: A medium suspected of containing a substance to be inspected is treated under a condit...
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JP3881165B2 |
To provide a method for producing a compound having high HIV activity. A process for the preparation of enantiomerically pure β-D-(-)- dxoxolane-nucleosides (e.g. a compound represented by formula 2 when thymine is used as a base) compr...
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