Document |
Document Title |
JPS6051474B2 |
The reaction of 1-(halo/cyano/sulfonyloxy)alkanoyl-2-(dibenzoxazepine-10-car
bonyl)hydr azines with an amine affords the corresponding 1-(substituted amino)alkanoyl-2-(dibenzoxazepine-10-carbonyl)hydrazines which compounds are useful ant...
|
JPS60184064A |
NEW MATERIAL:A phthalimide derivative shown by the formula I [R is H, or alkyl; ring A of broken line is group shown by the formula IVWVI; R1, R2, R4 and R5 are H, alkyl, or R1 and R2 or R4 and R5 are bonded to form a part of a ring of 3...
|
JPS6030313B2 |
|
JPS60123479A |
(57) [Abstract] Since this gazette is application data in front of an electronic application, the data of an abstract is not recorded.
|
JPS6016432B2 |
|
JPS60500176A |
(57) [Abstract] Since this gazette is application data in front of an electronic application, the data of an abstract is not recorded.
|
JPS59148768A |
NEW MATERIAL:A dibenzo[b,f][1,5]oxazocine derivative shown by the formula I (R1 and R2 are H, lower halogen, lower alkyl, trihalomethyl, lower alkoxy, or lower acryl; R3 is H, or lower alkyl, and R3 is H, or lower alkyl, and R3 and R4 ma...
|
JPS59130280A |
7-phenyl-7-phenoxymethyl-hexahydro-1,4-oxazepines of the formula I I wherein R1 is hydrogen, chlorine or methoxy and R2 is hydrogen or methyl, and their salts with physiologically tolerated acids, and their preparation, are described. Th...
|
JPS59128379A |
NEW MATERIAL:The compound of formula I (R1 and R2 are H, halogen, lower alkyl, trihalomethyl, lower alkoxy or lower acyl; m and n are integer of 1W4). EXAMPLE: 5H-Dibenzo[b,f][1,5]oxazocin-11(12H)one. USE: Intermediate of psychotropic ag...
|
JPS5993047A |
(57) [Abstract] Since this gazette is application data in front of an electronic application, the data of an abstract is not recorded.
|
JPS5993066A |
A method of counteracting the effects of histamine with aromatic azepinones and diazepinones and thiones thereof having the formula wherein: A is benzene, naphthalene, quinoline or pyridine; B is oxygen or sulfur: E is oxygen, sulfur or ...
|
JPS5914029B2 |
NEW MATERIAL:A compound I (R1,2 are lower alkyl, or together form a 5- or 6-membered ring; R3 is H, phenyl). EXAMPLE:6-Benzylidene-3,4-dimethyl-5,7-dioxo-2-phenyl-perhyd
ro-1,4-oxa zepin. USE:Central nervous system depressant. An interme...
|
JPS5912678B2 |
Compounds of the formula:
|
JPS5948450A |
Oxamic esters of the formulae I and II in which A and B denote hydrogen, chlorine, bromine or cyano and R<1> denotes an alkoxyethyl radical having 1 to 4 C atoms in the alkoxy radical, which can be used for the treatment of allergic dise...
|
JPS59508B2 |
Compounds of the formulae:
|
JPS5857431B2 |
Compounds of the formulae:
|
JPS58206520A |
PURPOSE: To provide the titled suppressing agent having low toxicity and exhibiting strong effect to inhibit the formation of metastatic nest, by using a specific dibenzooxazepine derivative. CONSTITUTION: The agent contains the compound...
|
JPS5840550B2 |
|
JPS5839145B2 |
2-[N-(2-Hydroxyethyl)-N-lower alkylamino methyl]-benzhydrols of formula in which R denotes a methyl or ethyl group, X denotes a fluorine, chlorine or bromine atom or a methyl group, Y denotes a fluorine or chlorine atom or a methyl or me...
|
JPS5817469B2 |
|
JPS5817470B2 |
|
JPS57501962A |
|
JPS57134483A |
Compounds of formula (I): (I) wherein: X is CH2, O, S or NR wherein R is hydrogen or C1-4 alkyl; Y and Z are independently selected from hydrogen, C1-4 alkyl, C1-4 alkoxy, halogen or CF3; R1 is hydrogen, C1-6 alkyl, phenyl or phenyl-C1-4...
|
JPS57128660A |
Aminoheterocycles of formula (I) and their acid addition salts are new (n is 1-3, A is nitrogen or CH. X is methylene, or provided A is not CH, also methyleneoxy. When A is CH, R is phenyl opt. 2-fluoro substd. and when A is N, R is phen...
|
JPS57106673A |
NEW MATERIAL:The compound of formulaI(R1 is H or lower alkyl; R2 is branched-chain lower alkyl; R3 is H, COOH, lower alkoxycarbonyl or lower alkoxy; R4 and R5 are lower alkyl, or R4 and R5 may together with N atom form a heterocyclic gro...
|
JPS57102877A |
Compounds are described of the formula (1) in which R1 is unsubstituted or substituted phenylalkyl, thienylalkyl or naphthylalkyl, or cinnamyl; R2 is a hydrogen atom, methyl or alkyl substituted by alkoxy or -COOH; W is alkylene; X is ci...
|
JPS5724356B1 |
1388582 Quinobenzoxazepine- and quinobenzothiazepine-derived amines E R SQUIBB & SONS Inc 5 June 1972 [24 June 1971] 26100/72 Heading C2C The invention comprises compounds of formulµ and their salts, wherein X, Y are each C 1-8 alkyl, a...
|
JPS5756449A |
A new class of chemical compounds and their process of preparation is described. These compounds have valuable properties as anti-secretory, anti-spasmodic, anti-ulcerogenic and anti-diarrheal agents.
|
JPS5735576A |
NEW MATERIAL:4,1-Benzoxazepin-3-acetic derivatives of formula I [R, R1 are H, lower alkyl, phenyl; R2 is H, halogen, lower alkyl which may be substituted with nitro or hydroxyl groups, aralkyl, formula II (n is 1W3; R5, R6 are lower alky...
|
JPS572278A |
NEW MATERIAL:A dibenzoxazepin derivative of formula I (R1 is H, 1W2 halogens, lower alkyl, or lower alkoxy; R2 is H or lower alkyl). EXAMPLE: 8-Ethoxycarbonyldibenzo[b,f][1,4]oxazepin-11(10H)one. USE: It has antilipemic activity, antiulc...
|
JPS56167622A |
NEW MATERIAL:Compounds of formula I (R1 is H, lower alkoxy; R2 is hydroxyl, lower alkoxy). EXAMPLE: 10, 11-Dihydro-4-methoxybenzo[ b, f ][ 1, 4 ]oxazepin-8-carboxylic ethyl ester. USE: Hypolipemic: they are used to prevent and treat vari...
|
JPS56167623A |
1. Anti-inflammatory compositions for local topical administration containing an effective amount of a compound of the general formula see diagramm : EP0039059,P10,F2 wherein X signifies a sulphur or oxygen atom, Y signifies the group -C...
|
JPS56166179A |
NEW MATERIAL:A dibenzoxazepine derivative shown by the formula I (R1 is H, halogen, or lower alkoxy; R2 and R3 are H, lower alkyl, or cycloalkyl). EXAMPLE: 10,11-Dihydro-4-methoxydibenzo[ b, f ][ 1, 4 ]oxazepine-8-carboxycyclohexylamide....
|
JPS56147778A |
NEW MATERIAL:A compound shown by the formula I [X is halogen, nitro; Y is phenyl, substituted phenyl, or pyridyl; A-B is a group shown by the formula II (Q is O, S, or hydrazono), formula III, formula IV (R1 is H, halogen, alkyl, etc.), ...
|
JPS56135487A |
1388582 Quinobenzoxazepine- and quinobenzothiazepine-derived amines E R SQUIBB & SONS Inc 5 June 1972 [24 June 1971] 26100/72 Heading C2C The invention comprises compounds of formulµ and their salts, wherein X, Y are each C 1-8 alkyl, a...
|
JPS565746B1 |
|
JPS5540855B2 |
A photographic light-sensitive material comprising a support having thereon at least one silver halide photographic emulsion layer and at least one of the layers of the photographic light-sensitive material containing a compound represen...
|
JPS5576869A |
NEW MATERIAL:A dibenzoxazepine derivative of formula I: (R1 is H, 1W2 halogens, lower alkyl, or lower alkoxy group; R2 is hydroxyl, lower alkoxy, or anilino group; R3 is H or acyl group). EXAMPLE: 10, 11-Dihydro-4-methoxy-dibenzo (b, f) ...
|
JPS558017B2 |
Hydrocurable compositions of a hydroxy(polyalkylenecarbonyloxy)alkyleneoxazolidine and a polyfunctional isocyanate are disclosed. The compositions are useful in forming films, paints, coatings, fibers, seamless flooring, coatings, impreg...
|
JPS5422978B2 |
The present invention relates to cyclopropylmethyl amines substituted by a heterocyclic radical.
|
JPS5498780A |
Polyfluorohydroxyisopropyl bicyclic and tricyclic carbostyrils, such as 2,3-dihydro-7-methyl-9-[2,2,2-trifluoro-1-hydroxy-1-(trifluo
romethyl)e thyl]-5H-pyrido[1,2,3-de]-1,4-benzoxazin-5-one, useful as antihypertensive agents.
|
JPS544955B2 |
The present invention relates to cyclopropylmethyl amines substituted by a heterocyclic radical.
|
JPS5427559A |
PURPOSE: Title compound of Formula I.
|
JPS53121782A |
PURPOSE: Decahydro-1,3-benzoxazepin-4-ones I(R1 is m-hydroxyphenyl or m-aralkyloxyphenyl; R2 is lower alkyl or aralkyl), e.g. 5a-(3-benzyloxyphenyl2,3,4,5,5a,6,7,8,9,9a-decahydro-3-methy
l-1,3-benzoxazepin-4-one.
|
JPS5335949B2 |
The present invention relates to cyclopropylmethyl amines substituted by a heterocyclic radical.
|
JPS5359697A |
Novel and biologically active tetracyclic compounds are disclosed of the formula: (I) or a pharmaceutically acceptable non-toxic salt thereof, wherein R1, R2, R3, and R4 are each hydrogen, hydroxy, C1-C6 alkyl, C1-C6 alkoxy, C1-C6 alkylt...
|
JPS5334791A |
|
JPS52128350A |
A new class of chemical compounds and their process of preparation is described. These compounds have valuable properties as anti-secretory, anti-spasmodic, anti-ulcerogenic and anti-diarrheal agents.
|
JPS52105184A |
PURPOSE: Morpholine derivatives I (R1 is H or lower alkyl; R2 is H, lower alkyl, lower alkenyl or aryl-lower-alkyl, etc.; A is lower alkylene; B is -CH2CH2-, -CH=CH-, etc.; C1 and C2 are 1,2-phenylene or substituted 1,2phenylene; D-E-is ...
|
JPS52100486A |
PURPOSE: -Glutamic acid N-carboxyanhydride of formula I.
|