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Matches 201 - 250 out of 14,059

Document Document Title
WO/2013/143259
The present invention relates to a phosphodiesterase-4 inhibitor capable of avoiding a vomit reaction. The phosphodiesterase-4 inhibitor is a compound, a prodrug or a solvate represented by DTPM. The name of DTPM is 1-(4-difluoro methoxy...  
WO/2013/147568
The present invention provides an aminostyrylbenzofuran compound of Formula (I), and a pharmaceutical composition comprising same. The pharmaceutical composition of the present invention comprising the compound of Formula (I), a pharmace...  
WO/2013/144097
The present invention relates to compounds of general formula I, (I), wherein the groups R1, R2 and m are defined as in claim 1, which have valuable pharmacological properties, in particular bind to the GPR40 receptor and modulate its ac...  
WO/2013/141523
The present invention relates to a method for preparing 5-acetoxymethylfurfural, comprising a step of synthesizing 5-acetoxymethylfurfural by reacting 5-halomethyl furfural with alkylammonium acetate. The present invention can provide a ...  
WO/2013/140969
The present invention is a photoresist composition which contains [A] a polymer that has a structural unit (I) containing an acid-cleavable group and a compound (I) that is represented by formula (1). In formula (1), each of R1, R2, R3 a...  
WO/2013/140946
Provided is a novel root parasitic plant germination inhibitor. Also provided is a root parasitic plant control agent comprising the root parasitic plant germination inhibitor. Further provided is a method for controlling a root parasiti...  
WO/2013/140506
Provided is a method for manufacturing 4,4'-oxydiphthalic acid with favorable productivity and high-yield via 4,4'-oxydiphthalonitrile, using 4-nitrophthalonitrile as a reaction raw material; the method including a hydrolysis step for hy...  
WO/2013/142873
The invention provides a novel, general, and facile strategy for the creation of small molecules with high structural and stereochemical complexity. Aspects of the methods include ring system distortion reactions that are systematically ...  
WO/2013/140347
Sulphonamide derivatives of benzylamine of formula (I), wherein A represents phenyl unsubstituted or substituted;or 9-or 10-membered bicyclic group, linked to –(O) x - (CH 2 ) y -through one of its aromatic carbon atoms,consisting of b...  
WO/2013/138243
The present disclosure encompasses bifunctional compounds resulting from the ring-expanding mono- and bis-carbonylation of glycidyl acrylates to afford the corresponding beta lactones and succinic anhydrides. Uses of the materials and po...  
WO/2013/138153
A process is disclosed for making dehydration products from an aqueous sugars solution including pentoses, hexoses or both, for example, an aqeous high fructose corn syrup solution, or from an aqueous solution of one or more of the alcoh...  
WO/2013/136294
A complex formed of at least one molecule of 5-(1,2-dihydroxy-ethyl) -3,4-dihydroxy-5H-furan-2-one or a derivative covalently bonded with at least one hydrocarbon radical with formula (A) as follows: wherein: • - m 1 = 1, 2, 3, 4, 5 or...  
WO/2013/138600
Radioprotector compounds including 3,3'-diindolylmethane (DIM) analogs, are provided. Further provided are methods for their use in reducing or preventing radiation damage, killing a tumor cell and protecting a non-tumor cell, and treati...  
WO/2013/136030
The present invention relates to powder compositions of a complex between an acid or a corresponding anion and at least one metal or corresponding metal cation, said corresponding anion or acid being selected from the group containing 2-...  
WO/2013/135869
The invention relates to a process for the preparation of optically active 1,2-diol of formula (S,S)-(I), or alternatively of formula (R,R)-(I) by asymmetric transfer hydrogenation of a compound of formula (II), or a compound of formula ...  
WO/2013/132262
The present invention is directed to new compounds of formula (I) as well as to pharmaceutically acceptable salts thereof, to a pharmaceutical composition comprising said compounds, and to the use of said compounds in therapy, and more p...  
WO/2013/133078
A polymer characterized by containing repeating units respectively represented by formulae [1a], [1b] and [1c]. The polymer enables the production of a single-layer-coated horizontally oriented film by a simple process. [In the formulae,...  
WO/2013/133208
The present invention is a method for producing a tetrahydrofuran compound represented by general formula (2), the method comprising a reaction step for bringing a furan compound represented by general formula (1) into contact with a pal...  
WO/2013/133489
A method for producing 5-hydroxymethyl-2-furfural (HMF) from maize syrup containing fructose comprises a conversion step in which a reaction product containing the 5-hydroxymethyl-2-furfural is produced by mixing and heating the maize sy...  
WO/2013/128378
The present invention relates to phenyl alkanoic acid derivatives (the compounds of Formula (I)); and their isotopic forms, stereoisomeric and tautomeric forms and mixtures thereof in all ratios, or pharmaceutically acceptable salts, pha...  
WO/2013/128294
The invention relates to a novel process for preparation of dronedarone of formula (I) and pharmaceutically acceptable salts thereof, characterized in that a compound of formula (II) - where L is leaving group - is reacted with compound ...  
WO/2013/128294
The invention relates to a novel process for preparation of dronedarone of formula (I) and pharmaceutically acceptable salts thereof, characterized in that a compound of formula (II) - where L is leaving group - is reacted with compound ...  
WO/2013/130958
The present invention relates to novel benzofuran-2-sulfonamide derivatives formula (I), processes for preparing them, pharmaceutical compositions containing them and their use as pharmaceuticals as modulators of chemokine receptors.  
WO/2013/124745
The invention relates to a novel process for the preparation of dronedarone (I) and pharmaceutically acceptable salts thereof (formula I), which comprises oxidizing a compound of formula (VI), or a salt thereof and the obtained product i...  
WO/2013/124745
The invention relates to a novel process for the preparation of dronedarone (I) and pharmaceutically acceptable salts thereof (formula I), which comprises oxidizing a compound of formula (VI), or a salt thereof and the obtained product i...  
WO/2013/125732
The present invention provides a compound having a GOAT inhibitory action, which is useful for the prophylaxis or treatment of obesity and the like, and has superior efficacy. The present invention is a compound represented by the formul...  
WO/2013/125211
The purpose of the present invention is to provide an optical film that produces a large amount of in-plane retardation and sufficient reverse wavelength dispersion even with a low film thickness. This optical film contains a thermoplast...  
WO/2013/125599
[Problem] To provide an organic compound which is easy to synthesize and has excellent chemical stability, semiconducting properties (high carrier mobility) and high solubility in a solvent. [Solution] A compound represented by formula (...  
WO/2013/122905
A method of making acid anhydrides from epoxide and carbon monoxide feedstocks is presented. In various aspects, the method includes steps of reacting the contents of a feed stream comprising an epoxide, a solvent, a carbonylation cataly...  
WO/2013/121235
The invention relates to a novel process for preparation of dronedarone of formula (I) and pharmaceutically acceptable salts thereof the hydroxyl group is removed, and the obtained product is isolated and, if desired, converted into a ph...  
WO/2013/121209
A compound of formula I, and its pharmaceutically acceptable salt or salts and physiologically hydrolysable derivatives in free form or salt form: (Formula (I)) wherein either Q1, CR6a and optionally R6b together form a cyclic moiety whe...  
WO/2013/121235
The invention relates to a process for preparation of dronedarone of formula (I) and pharmaceutically acceptable salts thereof characterized in that from the compound of formula (II). the hydroxyl group is removed,. and the obtained prod...  
WO/2013/120876
The present invention pertains to novel enaminoketones containing a CF3O-group, novel pyrazole-derivatives containing a CF3O group as well as to a novel process for their preparation comprising aminoformylation of CF30-ketones and cycliz...  
WO/2013/120229
Disclosed is a method for preparing aqueous nanoparticle suspensions of derivatives of 4,9-dihydroxy-naphtho[2,3-b]furan aliphatic acid esters. The compositions and the uses of the aqueous nanoparticle suspensions prepared according to t...  
WO/2013/121234
The invention relates to a novel process for the preparation of dronedarone (I) and pharmaceutically acceptable salts thereof which comprises oxidizing a compound of formula (IV) or a salt thereof with an oxidizing agent in an organic or...  
WO/2013/118847
An organic EL element with high efficiency and long life, an electronic device mounting said element, and compound making it possible to provide such an organic electroluminescent element are provided. Said compound is specifically repre...  
WO/2013/118907
An amide compound represented by formula (I) has an excellent pest control effect. (In the formula, Y represents a 3-7 membered saturated heterocyclic ring which contains, as ring-forming component(s), one or more atoms or groups that ar...  
WO/2013/118905
An amide compound represented by formula (I) has an excellent pest control effect. (In the formula, Y represents a 3-7 membered saturated heterocyclic ring which contains, as ring-forming component(s), one or more atoms or groups that ar...  
WO/2013/117120
Provided in the present invention are a 2-arylbenzofuran-7-formamide compound as shown in general formula I or a pharmacologically or physiologically acceptable salt thereof, a preparation method thereof and use thereof in preparing anti...  
WO/2013/117585
Disclosed is a method for obtaining furan derivatives from D-glucose. In said method, A) D-glucose is transformed into D-fructose in an enzymatic process in which redox cofactors are used and regenerated, one of the two redox cofactors b...  
WO/2013/114040
The present invention relates to novel organic compounds, to the process for synthesizing same and to the uses thereof, in particular in the field of cancer treatment. In particular, the present invention relates to novel anticancer comp...  
WO/2013/115378
The present invention relates to: a method for producing a ruthenium catalyst, wherein ruthenium supported by a metal oxide is pretreated with an aldehyde compound, a phosphorus compound and a lower alcohol compound; and a method for pro...  
WO/2013/110313
Compounds of formula (I) are provided wherein R1 represents H, CN and CF3; R2 represents 1-naphthyl, 3,5-dichlorophenyl, 4-(4-fluorophenylthio)phenyl or phenyl substituted with one or more substituent selected from halogen, methoxy, cyan...  
WO/2013/107904
The invention relates to an alkoxycarbonylation process for the preparation of an optionally substituted alkanoic acid ester comprising reacting: (a) an optionally substituted alkene or a mixture thereof; (b) a source of a group 8-10 met...  
WO/2013/107947
The present invention describes a method for pretreating lignocellulosic biomass comprising: a) a step of acid hydrolysis of the biomass with an acid solution resulting in a liquid fraction and a solid fraction, b) a step of separating t...  
WO/2013/109477
Processes are disclosed for the conversion of a carbohydrate source to hexamethylenediamine (HMDA) and to intermediates useful for the production of hexamethylenediamine and other industrial chemicals. HMDA is produced by direct reductio...  
WO/2013/107948
The present invention relates to a method for preprocessing lignocellulosic biomass, include: a) a step for the acid hydrolysis of the biomass using an acid solution so as to obtain a liquid fraction and a solid fraction; a step of separ...  
WO/2013/105118
Disclosed herein is a novel route of synthesis of syn azide epoxide of formu 5, which is used as a common intermdeiate for asymmetric synthesis of HIV protease inhibitors such as Amprenavir, Fosamprenavir, Saquinavir and formal synthesis...  
WO/2013/105708
The present invention relates to a method for preparing α-metylene lactone comprising the steps of: (A) preparing an enolate intermediate by reacting lactone with alkyl formate under conditions in which an alcoxide base exists; and (B) ...  
WO/2013/105118
Disclosed herein is a novel route of synthesis of syn azide epoxide of formu 5, which is used as a common intermdeiate for asymmetric synthesis of HIV protease inhibitors such as Amprenavir, Fosamprenavir, Saquinavir and formal synthesis...  

Matches 201 - 250 out of 14,059