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JPH10279583A |
To obtain a new heterotricyclic herbicide comprising a specific heterotricyclic compound, its N-oxide or an agrichemically suitable salt thereof and useful as an inexpensive, low-toxic and environmentally safe herbicide for controlling u...
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JPH10279578A |
To produce the subject new compound usable for treating disorders associated with dysfunction in serotoninergic transmission, e.g. mental disorders or retrogressive diseases. This N-arylpiperidine compound is represented by formula I [(m...
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JPH10509706A |
A compound of formula (I), in which: R1 is lower alkyl, cyclo(lower)alkyl, optionally substituted aryl, optionally substituted heterocyclic group, cyclo(lower)alkyl(lower)alkyl, or ar(lower)alkyl; R2 is hydrogen, hydroxy or protected hyd...
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JPH10237071A |
To obtain a new compound which exits in a form of racemic mixture or optical isomer and is useful for treatment of disorders in which involvement of serotoninergic system is confirmed, e.g. mental disorders, etc. This compound is represe...
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JP2776906B2 |
Aminomethylheterocyclic compounds of the formula (I) in which X, R, R<1> and R<2> have diverse meanings, the acid addition salts thereof, the use thereof in pesticides and heterocyclic intermediates. The aminomethylheterocyclic compo...
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JPH10167964A |
To obtain the subject composition that contains a novel coumarin derivative as an active ingredient and is useful for treatment or prevention of diabetes as a hypoglycemic. The objective composition contains, as an active ingredient, abo...
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JPH10505847A |
The invention relates to new substituted pyrazol derivatives of general formula (I) in which: R1, R2, R3, R4, R5 and R6 have the meanings given in the description, agents with herbicidal action containing at least one compound of formula...
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JP2753622B2 |
This invention relates to carbostyril derivatives represented by general formula (1), a process for their preparation, and an agent for inhibiting agglutination of platelets containing them as an active ingredient, wherein A represents a...
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JPH10130267A |
To obtain the subject compound useful for a herbicide, having no phytotoxicity to cultivated plants, capable of destroying various kinds of weeds once with a small amount, by converting a carbon atom at the 4-position of a thiochroman in...
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JP2738010B2 |
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JPH1087668A |
To obtain a new coumarin quinolone carboxylic acid (salt) capable of inhibiting the growth of cells of breast cancer, spleen cancer, pharyngeal cancer, etc., and useful as an antibacterial agent, an antitumor agent and an antiviral agent...
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JPH10501001A |
Novel imidazole derivatives as histamine receptor H3 antagonists and/or agonists, preparation thereof and therapeutical uses thereof. Chemical compounds for use as histamine receptor H3 agonists, partial agonists or antagonists, having g...
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JPH10500673A |
3-Phenylpyrazoles (I) are new. In (I), R1 is e.g. H, CN, NO2, halo, Hc opt. substd. by halo, CN-1-4C alkyl, 1-8C alkyl-OCOR6, Hc-Z-R6, ZR6, SO2Cl, SO2OR6 etc.; R2 is CN, CF3 or halo; R3 is H or 1-4C alkyl opt. substd. by halo; R4 = 1-4C ...
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JPH107659A |
To obtain the subject compound having strong effects against resistant insect pest and properties giving no harmful influence to men and beasts and the environment and extraordinary excellent insecticidal activities as an effective ingre...
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JPH09512526A |
This invention relates to single enantiomers of novel cis-substituted 1,3-oxathiolanes, of formula (I) wherein R1 is hydrogen, and R2 is cytosine or 5-fluorocytosine, and pharmaceutically acceptable salts and esters thereof. This inventi...
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JPH09323991A |
To obtain the subject new derivative useful as a treating agent for hypertension, heart failure, nephritis, etc., an intraocular pressure lowing drug, etc., by reacting a specific carboxymethylidenecycloheptoimidazole derivative with a d...
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JP2690480B2 |
To obtain the subject novel compound that is useful as a synthetic intermediate for herbicide. This novel compound is 4-formyltetrahydropyran that is represented by formula I (R1 is H, a 4-12C alkyl, a 4-12C cycloalkyl, an aryl, a hetero...
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JP2659863B2 |
Use of a compound of formula (I) or a pharmaceutically acceptable derivative thereof in the manufacture of a medicament for the treatment of hepatitis B is disclosed.
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JP2656383B2 |
PCT No. PCT/KR92/00007 Sec. 371 Date Dec. 9, 1993 Sec. 102(e) Date Dec. 9, 1993 PCT Filed Mar. 9, 1992 PCT Pub. No. WO92/15568 PCT Pub. Date Sep. 17, 1992.The present invention relates to novel benzenesulfonylurea derivatives, having a h...
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JP2644357B2 |
Disclosed are compounds of the formula wherein R1 is hydrogen; R2 is a purine or pyrimidine base or an analogue or derivative thereof; Z is S, S=O or SO2; and pharmaceutically acceptable derivatives thereof. Also described are use of the...
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JPH09176158A |
To obtain a new nitrogen-containing heterocyclic compound high in light absorbance and useful for dyestuffs, additives, medicines, agrochemicals, etc. This compound is expressed by formula I [R1-R6 are each H, a substituent; Y1 is O, S, ...
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JP2602931B2 |
The present invention involves compounds having the structure: (a) -A- is selected from the group consisting of -CH2-, - @@-, and -@-; (b) -Y is selected from certain low molecular weight alkyl chains which terminate in specific unsatura...
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JP2601566B2 |
Benzamide piperidinyl cpds. of formula (I) and their salts N-oxides and isomers are new. A = CH2-CH2-, -CH2-CH2-CH2- or -(CH2)4- where 1 or 2 H of these radicals may be replaced by 1-6C alkyl. R1 = H or halo. R2 = H, NH2, mono- or di(1-6...
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JPH09502453A |
PCT No. PCT/FR95/00683 Sec. 371 Date Jan. 19, 1996 Sec. 102(e) Date Jan. 19, 1996 PCT Filed May 24, 1995 PCT Pub. No. WO95/32200 PCT Pub. Date Nov. 30, 1995The present invention pertains to the field of organic chemistry, and particularl...
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JPH09502178A |
PCT No. PCT/EP94/02821 Sec. 371 Date Feb. 15, 1996 Sec. 102(e) Date Feb. 15, 1996 PCT Filed Aug. 25, 1994 PCT Pub. No. WO95/06641 PCT Pub. Date Mar. 9, 1995Substituted 1-amino-3-phenyluracils I I where the variables have the following me...
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JPH08333367A |
PURPOSE: To obtain a new oxathiolane derivative having excellent antifungal action and effective against fungal diseases of man and animal. CONSTITUTION: This oxathiolane derivative is a compound expressed by formula I (Ar1 is phenyl sub...
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JPH08319285A |
To provide a novel substituted pyridne that is a specific 2,6-substituted pyridine carboxylic derivative, can control undesirable plants, when an effective amount of this compound is applied to the plant sites and is useful as a herbicid...
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JP2556524B2 |
4-Formyltetrahydropyrans of the general formula I (I) where R1 is hydrogen, C1-C12-alkyl, C2-C12-alkenyl, C1-C6-alkoxy-substituted C1-C12-alkyl, C4-C12-cycloalkyl, unsubstituted or substituted aryl, hetaryl or aralkyl, or an unsubstitute...
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JP2531935B2 |
PURPOSE: To obtain the subject compound for e.g. the treatment of infections caused by retroviruses such as HIV industrially advantageously by, for example, a process comprising deductively aminating an isoindol-2-yl-containing α- hydro...
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JPH08217774A |
PURPOSE: To obtain a new type carbonate or a dithiocarbonate compound available from a fish oil highly unsaturated fatty acid, etc., conventionally having no suitable use, etc. CONSTITUTION: This heterocyclic compound is represented by t...
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JPH08507758A |
Compounds of formula X-NH-CO-Z and pharmaceutically acceptable salts thereof, and the use of a compound of said formula or a pharmaceutically salt thereof, wherein X is a monocyclic or polycyclic aromatic group, Z is of sub-formula (h), ...
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JPH08506334A |
Heterocyclic aminomethyl-4 piperidine derivatives corresponding to general formula (1), and the therapeutically acceptable salts of these molecules. The invention also concerns the use of compounds of general formula (1) in therapy and p...
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JPH07121941B2 |
This invention relates to certain quinolinyl-benzoheterobicyclic compounds and their use as valuable pharmaceutical agents, particularly as lipoxygenase inhibitors and/or leukotriene antagonists and/or as mediator release inhibitors usef...
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JPH07252149A |
PURPOSE: To obtain an ophthalmic medicine containing a 1,5-benzoxathiepin derivative, exhibiting an excellent local action, reduced in side effect and excellent in safety. CONSTITUTION: This ophthalmic medicine contains a compound of the...
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JPH07507002A |
A catalyst solution comprising one or more compounds of a metal catalyst and an organic solvent selected from the group consisting of a glycol derivative, an alkyl pyrrolidone, and an alkoxy ethyl ether, wherein no additional chloride-co...
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JPH07196651A |
PURPOSE: To provide a new compound having excellent herbicide effect, plant growth controlling effect, and selectivity, useful as a herbicide and a plant growth controlling agent. CONSTITUTION: This compound is a compound represented by ...
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JPH07188223A |
PURPOSE: To obtain a new oxathiane derivative or its salt having a higher safety and a stronger wide-ranging antifungal activity and useful as an antifungal agent. CONSTITUTION: An oxathiane derivative is represented by formula I {ph is ...
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JPH07188219A |
PURPOSE: To obtain a cyclic acetal which itself exerts a good herbicidal effect and is useful as an intermediate for preparation of a substituted salicylic acid derivative having a good herbicidal effect and/or bioregulatory activity. CO...
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JPH07133275A |
PURPOSE: To provide a novel compound which exhibits inhibitory activities against biosynthesis of leucotriene and is useful for the treatment of allergic symptoms and various kinds of inflammatory symptoms. CONSTITUTION: There is provide...
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JPH07109221A |
PURPOSE: To obtain a mutation inducing HIV-RT inhibitor useful for improving or maintaining antiviral receptivity to zidovudine of HIV population. CONSTITUTION: This mutation inducing inhibitor of a human immunodeficiency virus reverse t...
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JPH0735368B2 |
2-(8-Azabicyclo[3.2.1]oct-8-yl)alkanols of the formula (I) wherein Q is S or CH=CH; X is H, OH or another aromatic substituent; R is hydrogen, alkyl, alkenyl or alkynyl; Y and Y1 are taken together and are arylmethylene or aralkylmethyle...
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JPH0735380B2 |
Disclosed herein are 2- or 6-fluoromethyl-3-pyridinecarboxylate derivatives with 5-[(heterocyclic)ylidene]amino substitution useful as herbicides and herbicide intermediates.
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JPH0723365B2 |
PCT No. PCT/SE86/00038 Sec. 371 Date Nov. 26, 1986 Sec. 102(e) Date Nov. 26, 1986 PCT Filed Jan. 31, 1986 PCT Pub. No. WO86/04584 PCT Pub. Date Aug. 14, 1986.Novel compounds of formula (I), wherein R1 is selected from hydrogen, halogen; ...
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JPH0714928B2 |
The invention relates to N-phenylsulfonyl-N'-pyrimidinylureas and N-phenylsulfonyl-N-triazinylureas of the general formula (I) wherein Q is selected from a radical +TR Z is oxygen or sulfur, E is nitrogen or =CH-, R2 is hydrogen, C1-C4 a...
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JPH0725857A |
PURPOSE: A obtain a new condensed heterocyclic derivative showing herbicidal activity against gramineous and non-gramineous weeds without damaging crops in water treatment in paddy field, soil treatment in upland farming and foliar treat...
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JPH075567B2 |
1,3-Benzodioxoles and 1,3-benzodithioles substituted with a 6-fused imidazole of Formula I which are useful as angiotensin II antagonists.
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JPH075590B2 |
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JPH07613B2 |
NEW MATERIAL:A compound expressed by formula I (R<1> is H or alkyl, m is 2, 3 or 4; R<2> is H, alkyl, halogen, nitro, cyano, alkoxy, alkylthio, amino, acyl, etc.; l is 1, 2, 3, 4, 5, 6, 7 or 8; X, Y, W and Z are c, O, S or N, provided th...
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JPH07618B2 |
The present invention relates to a method of preparing BCH-189 and various analogues of BCH-189 from inexpensive precursors with the option of introducing functionality as needed. This synthetic route allows the stereoselective preparati...
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JPH072844A |
PURPOSE: To obtain a new saturated heterocyclic carboxylic acid amide which is useful as a prophylactic and/or therapeutic agent for diseases caused by PAF because of its PAF antagonistic action. CONSTITUTION: A compound of the formula I...
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