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WO/1993/011759A1 |
This invention relates to novel diaminoalkanoic acid derivatives that inhibit platelet aggregation and thrombus formation in mammalian blood thereby being useful in the prevention and treatment of thrombosis associated with disease state...
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WO/1993/011118A1 |
Herbicidal compounds of formula (I) where: Az is imidazol-1-yl or 1,2,4-triazol-1-yl; each X represents halogen, carboxy, nitro, cyano, a group COR5, COOR5 or S(O)pR5, or an optionally substituted alkyl, alkoxy, aryl or heteroaryl group;...
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WO/1993/011124A1 |
The pyrrole derivatives having general formula (1), wherein X and X' represent H, alkyl, alkoxy, halogen, nitro, amino, and R is H, alkyl, aryl, arylalkyl, cycloalkylmethyl, are active against pathogenic microorganisms, and particularly ...
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WO/1993/010103A1 |
The invention embraces compounds of formula (I) and salts thereof, wherein: X and Y are independently selected from various optionally substituted alkoxy, alkenyloxy, alkynyoxy and phenoxy groups; W is oxygen or sulfur; R1 is hydrogen or...
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WO/1993/010101A1 |
Benzimidazole anthelmintic agents of the formula (I) and their non-toxic salts, wherein R1, which is in the 5(6)-position,is either H or certain stated substituents, "alk" is a methylene or ethylene group; R2 is cyano, C2-C4 alkenyl, C2-...
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WO/1993/009114A1 |
An antifungal compound represented by formula (I), wherein X is independently both F or both Cl or one X is F and the other is Cl; Y = (a), (b), (c), (d), (e), (f) or (g); R' = (C¿1?-C¿10?)alkyl, (C¿2?-C¿10?)alkenyl, (C¿2?-C¿10?)al...
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WO/1993/009100A1 |
Herbicidal triazolecarboxamides are useful as agricultural chemicals. In particular the compounds are useful as herbicides, both general and selective, both post-emergent and pre-emergent. Examples of selective activity include excellent...
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WO/1993/008153A1 |
Cyclohexenone derivates have the formula (I), in which R?1¿ stands for alkyl, alkenyl, alkinyl, cycloalkyl, aloxyalkyl, alkylthioalkyl, possibly substituted phenyl, possibly substituted benzyl, possibly substituted 5-/6-membered heteroa...
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WO/1993/008162A1 |
The present invention is directed to a compound of formula (I), wherein R represents a hydrogen atom or an acyl, aroyl or cycloalkylcarbonyl radical or a residue of formula (Ia); R1 represents an alkyl radical; R2 represents an aryl or h...
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WO/1993/008361A1 |
A highly efficient anti-explosion pad (6, 7) comprising multiple sheets of expanded metal net (10) separated by a core layer of porous material such as fiberglass, cotton batting or an assembly of miniature balls (22, 23, 24) formed from...
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WO/1993/007138A1 |
A compound represented by general formula (I), which has an agrohorticultural bactericidal activity, wherein Q represents (a) or (b); Y represents CR?6¿ or N; A represents an optionally substituted aryl or heterocyclic group; and B repr...
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WO/1993/007534A1 |
A photographic element comprising a support, at least one photosensitive silver halide layer and associated therewith a colour coupler of general formula (1) or (2), wherein A and B represent the same or different electron-withdrawing gr...
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WO/1993/007139A1 |
The invention provides antifungal compounds of formula (I) and the pharmaceutically acceptable salts thereof, wherein R is phenyl substituted by up to 3 substituents each independently selected from halo and trifluoromethyl; R1 is C1-C4 ...
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WO/1993/007124A1 |
A nitrogenous heterocyclic compound represented by general formula (I) or a pharmacologically acceptable salt thereof, efficacious in treating various ischemic cardiac diseases, wherein ring A represents a benzene, pyridine or cyclohexan...
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WO/1993/005048A2 |
Substituted sulphonyl ureas have the general formula (I), in which n and m equal 0 or 1 and the substituents have the following meaning: R?1¿ is hydrogen, alkyl, alkenyl or alkinyl; R?2¿ is halogen or trifluoromethyl, when m equals 0 o...
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WO/1993/005027A1 |
A triazolylated tertiary amine compound represented by general formula (I) or a salt thereof, having an aromatase inhibitory activity and being useful for preventing and treating breast cancer, mastopathy, endometriosis, prostatomegaly, ...
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WO/1993/005020A1 |
Novel indole compounds inhibit HIV reverse transcriptase, and are useful in the prevention or treatment of infection by HIV and the treatment of AIDS, either as compounds, pharmaceutically acceptable salts, pharmaceutical composition ing...
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WO/1993/004042A1 |
A carbostyril derivative represented by general formula (I), useful as a platelet agglutination inhibitor, wherein A represents lower alkylene; RA represents -NR1R2, wherein R1 represents lower alkyl substituted with lower alkoxycarbonyl...
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WO/1993/004043A1 |
Compounds of formula (I) wherein Ar, W, Z, Q, R1, U, and T are as set forth herein, are described. These compounds are active as agents against retroviruses and in particular against HIV.
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WO/1993/002058A1 |
A benzimidazole anthelmintic agent of formula (I) or a non-toxic salt thereof, wherein R1, which is in the 5- or 6- position, is either (i) benzoyl, phenyloxy, phenylthio, phenylsulfinyl, phenylsulfonyl, phenylsulfonyloxy, C1-C6 alkyl, C...
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WO/1993/002059A1 |
A benzimidazole derivative of formulae (IA) or (IB) or a non-toxic salt thereof, wherein R, which in the compounds (IA) is in the 5- or 6-position, is either (i) H, benzoyl, phenyloxy, phenylthio, phenylsulfinyl, phenylsulfonyl, phenylsu...
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WO1993002062A1 |
A piperazine derivative represented by general formula (I) and a salt thereof, wherein B represents phenyl or pyridyl; m represents an integer of 2 or 3; p represents an integer of 1 or 2; R<1> represents hydrogen or halogen; and A repre...
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WO/1993/001183A1 |
The enantiomer of 2-[5-(3,5-dimethylpyrazol-1-yl)pentylsulphinyl]-4,5-diphenyl
imidazole which, in dilute solution in dichloromethane at room temperature, rotates plane-polarised light of the sodium D wavelength to the right, or a pharma...
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WO/1993/000336A1 |
An iminosulfonylurea derivative represented by general formula (1) or salts thereof, a herbicide containing said derivative, and a method for killing weeds or inhibiting the growth thereof by applying said derivative, wherein Q represent...
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WO/1992/022313A1 |
A renin inhibiting compound of formula (I), wherein R�0? is a mimic of the Phe-His dipeptide sequence of angiotensinogen which precedes the renin cleavage site; R�4? is loweralkyl, cycloalkylalkyl or arylalkyl; R�5? is hydrogen, lo...
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WO/1992/022536A1 |
The invention concerns vinylimidazoles, vinyltriazoles and vinyltetrazoles of general formula (I) with a bicyclic substituent group. Such compounds have an enhanced aromatase-inhibiting action.
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WO/1992/021648A1 |
The present invention relates to compounds of formula (I).
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WO/1992/020674A1 |
The invention provides compounds of general formula (I), or a physiologically acceptable salt, solvate or metabolically labile ester thereof wherein R1 represents a hydrogen atom or a halogen atom or a group selected from C1-6alkyl, C2-6...
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WO/1992/020642A1 |
This invention relates to bis mono- and/or bicyclic aryl and/or heteroaryl compounds exhibiting protein tyrosine kinase inhibition activity. More specifically, it relates to the method of inhibiting abnormal cell proliferation in a patie...
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WO/1992/020659A1 |
Substituted pyridines having at the 3 or 5 position a carbonyl oxy(thio)ester or a heterocyclocarbonyl and at the other a substituted alkyl group, herbicidal compositions and methods of use thereof.
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WO/1992/020711A2 |
The invention concerns LHRH antagonists of the general formula (I), in which X is an acyl group, X�1? is a D-Nal, X�2? is D-(4-Cl)-Phe, X�3? is D-(3)-Pal, X�6? is D-Cit or D-Neu, X�8? is L-Arg or L-Neu, at least one of the grou...
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WO/1992/019600A1 |
A process for the production of N-acylimidazoles by the reaction of a carboxylic anhydride with carbonyldiimidazole is disclosed. The products are useful as chemical intermediates.
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WO/1992/018463A1 |
Specified cinnamic acid derivatives, such as methyl 4-(4-acetoxy-3-methoxycinnamamide)-1-methyl-1-cyclohexanecar
boxylate, and pharmaceutically acceptable salts thereof, which are useful as an allergy type IV reaction inhibitor.
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WO/1992/018092A2 |
A class of 1-arylheteroarylalkyl substituted-1H-1,2,4-triazole compounds is described for use in treatment of circulatory disorders such as hypertension. Compounds of particular interest are angiotensin II antagonists of the formula (I) ...
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WO/1992/017451A1 |
Compounds of formula (I) or a biolabile ester thereof, or a pharmaceutically acceptable salt of either, wherein R1, R2, R3 and R4 are each independently selected from H or C1-C4 alkyl; R5is (CH2)mSO2R6, (CH2)mNHSO2R6 or (CH2)mNHCOR7; R6 ...
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WO/1992/017472A1 |
The description relates to novel compounds of the general formula (I) in which R in position 3 or 4 represents hydrogen, methyl, chlorine or bromine and R?2� is C�1?C�100?-alkyl, C�3?-C�7?-cycloalkyl or benzyl, and their pharma...
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WO/1992/017474A1 |
The invention provides antifungal compounds of formula (I) and pharmaceutically acceptable salts thereof, wherein R is phenyl optionally substituted by 1 to 3 substituents each independently selected from halo and CF3; R1 is C1-C4 alkyl;...
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WO/1992/017470A1 |
Imidazole derivatives of formula (I), wherein R1 represents optionally substituted phenyl, R2 represents alkyl optionally substituted by hydroxy, X1 represents a bond, oxygen, -S(O)n-, -CH2O- or - CH2N(R6)-, wherein n is 0, 1 or 2 and R6...
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WO/1992/017176A1 |
Compounds are disclosed which are retroviral protease inhibitors. Also disclosed are methods of using the compounds and compositions for inhibiting a retroviral protease and for treating an HIV infection.
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WO/1992/016525A1 |
The present invention relates to novel thiophenesulfonylurea derivatives having a herbicidal activity, which is described in general formula (I), wherein P is P-1, P-2 or P-3 , wherein R is (1), (2), (3), wherein a is O or S; R2 is C1-C6...
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WO/1992/016522A1 |
N-pyridinesulfonyl-N'-pyrimidinyl- and -triazinyl-ureas of formula (I), wherein R1 is hydrogen or fluorine; or R1 together with R3 is a C2-C4alkylene chain; R3 is hydrogen, fluorine or C1-C3alkyl; R2 is hydrogen, fluorine or C1-C3alkyl; ...
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WO/1992/015576A1 |
A pyridine sulfonylurea herbicide, composition thereof and a method for its use that results in the control of blackgrass in cereal crops and general control of all plant growth.
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WO/1992/015568A1 |
The present invention relates to novel benzenesulfonylurea derivatives, having a herbicidal activity, which is described in the structure of general formula (I), wherein R1 is H, C1-C3 alkyl, C1-C3 haloalkyl, halogen, CN, NO2, C1-C3 alko...
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WO/1992/015578A1 |
The invention concerns triheteroarylmethanes of general formula (I), where R stands for a cyano or CH�3? group, a fluorine, chlorine or bromine atom, an alkoxyimino residue -CH=N-OR' or an acide amide residue -C(O)NR'R'', where R' and ...
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WO/1992/014728A1 |
The present invention relates to novel pyridine sulfonyl urea derivatives, having a herbicidal activity, which is described in structure of general formula (I), wherein P is P-1, P-2, P-3 or P-4; E is single bond or CH2; R2 is C1-C6 alky...
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WO/1992/014703A1 |
A process for transforming a carbonyl compound into its corresponding epoxide, which comprises contacting the carbonyl compound with either trimethylsulphonium hydrogen sulphate and/or bis(trimethylsulphonium) sulphate or trimethylsulpho...
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WO/1992/014715A1 |
The invention concerns sulfonyl urea derivatives of formula (I), wherein R?1� stands for optionally substituted alkyl or phenyl; alkenyl or propargyl; alkylamino or dialkylamino; R?2� stands for hydrogen, halogen, optionally halogen-...
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WO/1992/013845A1 |
The invention concerns new herbicidal and plant-growth regulation compounds of formula (I), in which Q, W, R?1�, R?2�, R?3�, Y and Z as shown in formula (I) are as defined in claim 1, as well as salts of these compounds. They can b...
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WO/1992/013830A1 |
Fungicidal compounds having formula (I) and stereoisomers thereof, wherein A is hydrogen, halo, hydroxy, C1-4 alkyl, C1-4 alkoxy, C1-4 haloalkyl, C1-4 haloalkoxy, C1-4 alkylcarbonyl, C1-4 alkoxycarbonyl, phenoxy, nitro or cyano; R1 and R...
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WO/1992/013798A1 |
Solid peroxyacid bleach precursor compositions are provided in which the external surfaces of a particulate peroxyacid precursor material is treated with from 2 % to 20 % by weight of a solid organic acid compound of Mpt > 30 �C and an...
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