Heterocyclic Compounds

Matches 1,201 - 1,250 out of 5,408	< 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 >

Document	Document Title
WO/1994/027976A1	TRIAZOLE DERIVATIVE OR SALT THEREOF, AND FUNGICIDE CONTAINING THE SAME A triazole derivative represented by general formula (1) or a salt thereof, and a fungicide containing the same, wherein R1 and R2 represent each methyl, or R1 and R2 are combined together to represent ethylene. The compound (1) has a hi...
WO/1994/026700A1	O-BENZYL OXIME ETHER DERIVATIVES AND THEIR USE AS PESTICIDES Compounds of formula (I) in which Y is hydrogen, C1-C4alkyl, C1-C4alkoxy, OH, CN, NO2, Si(CH3)3, CF3 or halogen, Z is a group (a) or (b) and R1 is hydrogen, C1-C4alkyl, C2-C4alkenyl, C2-C4-alkynyl, C3-C6cycloalkyl, phenyl which is unsubs...
WO/1994/026734A1	AZOLYLAMINE DERIVATIVE An antifungal agent containing as the active ingredient a compound represented by general formula (I) or an acid-addition salt thereof, in particular, one having an absolute configuration of (R, R) at the asymmetric carbon atoms or an ac...
WO/1994/026737A1	IMIDAZOLYLQUINOXALINEDIONE DERIVATIVE AND PHARMACEUTICAL COMPOSITION THEREOF An imidazolylquinoxalinedione derivative, represented by general formula (I), useful as a glutamate receptor antagonist, a pharmaceutically acceptable salt thereof, and a pharmaceutical composition containing the same as the active ingre...
WO/1994/026709A1	GUANIDINE DERIVATIVES AS INHIBITORS OF Na+/H+ EXCHANGE IN CELLS Guanidine derivatives of formula (I), wherein Y is N or C-R1 (in which R1 is hydrogen, lower alkyl, hydroxy, protected hydroxy, etc.), R2 is hydrogen, aryl which may have one suitable substituent, aryloxy, etc., R3 is hydrogen, lower alk...
WO/1994/025452A1	PROCESS FOR PREPARING INTERMEDIATES FOR THE SYNTHESIS OF ANTIFUNGAL AGENTS Disclosed is a process for preparing chiral compounds of formula (I) wherein: X1 and X2 are independently F or Cl; and E is -SO2R2, wherein R2 is C1-C6 alkyl, -C6H4CH3 or -CF3; its enantiomer and racemates thereof, useful in the synthesi...
WO/1994/025665A1	RADIATION-INDUCED FIXATION OF DYES A process for dyeing or printing organic material, preferably fibre material, which comprises applying dyes together with a colourless cationic compound containing at least two polymerisable double bonds, as well as additional optional a...
WO/1994/025469A1	QUINOXALINDIONE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN DRUGS Described are compounds of formula (I) in which R1, R5, R6, R7 and R8 are as defined in the application, plus their preparation and their use in drugs.
WO/1994/024868A1	NEMATICIDAL AGENTS BASED ON 2-DICHLOROMETHYL-1,3,4-OXADIAZOLES The invention concerns the use, as insecticides, nematicides and acaricides, of 2-dichloromethyl-1,3,4-oxydiazoles, some of them prior art compounds, of general formula (I) in which X is a single bond or one of the following groups: -O-,...
WO/1994/024305A1	CHIRAL SYNTHESIS OF TERTIARY ALCOHOLS WITH A HYDROLASE Method of preparing an optically active compound of formula (I), wherein R and R1 are independently alkyl, alkenyl, alkynyl, alkoxy, alkoxyalkyl, cycloalkyl, aryl, aralkyl, a heterocyclic group or a C1-C4 alkyl-heterocycle, each being op...
WO/1994/023577A1	TRIAZOLYL AND TETRAZOLYL PHENYL SUBSTITUTED CARBAPENEM COMPOUNDS Triazolyl and tetrazolyl phenyl substituted carbapenems of formula (I) are disclosed. One or two of the variables X, Y and Z represent nitrogen atoms. The heteroaryl ring may be charged or uncharged. Pharmaceutical compositions and metho...
WO/1994/022812A1	IMINO-SUBSTITUTED PHENYLACETIC ACID AMIDES, THEIR PREPARATION AND FUNGICIDES CONTAINING THEM Described are compounds of the formula (I) in which Y is oxygen or an NR6 group; Z1 and Z2 are hydrogen, halogen, alkyl, alkenyl, alkinyl, alkoxy, alkenyloxy, haloalkyl, haloalkoxy, haloalkenyloxy, cyano or nitro; R1 is hydrogen, alkyl, ...
WO/1994/022413A2	TRIAZOLE SUBSTITUTED QUINOLINE DERIVATIVES The invention relates to pharmaceutical compositions for the treatment or prevention of lesions of gastrointestinal mucous membranes and having secretion inhibiting, cytoprotective activities. The compositions contain in a biologically e...
WO/1994/022852A1	QUINOLINES AS TYPE IV PHOSPHODIESTERASE INHIBITORS Optionally 6,8-substituted quinolines of formula (I) wherein: R1 is selected from hydrogen; lower alkyl; cycloalkyl; cycloalkyloxy; cycloalkylamino; cycloalkyl lower alkyl; lower alkoxy; formyl; hydroxy-lower alkyl; carboxyalkyl; optiona...
WO/1994/022855A1	NITROGEN-CONTAINING FUSED-HETEROCYCLE COMPOUNDS The present invention relates to a nitrogen-containing heterocyclic compound exhibiting an inhibitory activity against cGMP-PDE. The compound represented by formula (I) or a pharmacologically acceptable salt thereof, wherein R1 represent...
WO/1994/022826A1	PERIPHERAL VASODILATING AGENT CONTAINING N-ACYLATED 4-AMINO PIPERIDINE DERIVATIVES AS ACTIVE INGREDIENTS The present invention relates to novel peripheral vasodilating agents characterized by each containing as an active ingredient, a piperidine derivative or pharmaceutically acceptable salt thereof having excellent peripheral vasodilating ...
WO/1994/022835A2	HETEROCYCLIC COMPOUNDS AS PLATELET AGGREGATION INHIBITORS A compound of the general formula (I): (M1)n-Q-(M2)1-n-L-A wherein: n is 0 or 1; M1 is an amino group; Q is an aromatic heterocyclic group containing a basic nitrogen atom; M2 is an imino group; L is a template group; and A is an acidic ...
WO/1994/022842A1	1-AMINO-3-PHENOXY PROPANE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE This invention relates to 1-amino-3-phenoxy-propane-derivatives of formula (1) (in which A, B, R, Rx, X and Z are defined as in the specification described) and methods for their preparation. These compounds may be used as modulators of ...
WO/1994/021606A1	PENTAFLUOROSULPHANYLPHENYL AND PENTAFLUOROSULPHANYLPYRIDIL SUBSTITUTED HETEROAROMATIC COMPOUNDS WITH INSECTICIDAL OR ACARICIDAL ACTIVITY Compounds with insecticidal or acaricidal activity have formula (IA) or (IB), wherein Ra represents hydrogen or from 1 to 4 optional substituents and Rb represents from 1 to 3 optional substituents and wherein A represents an optionally ...
WO/1994/019346A1	SUBSTITUTED HETEROARYLALKYLTHIOPYRIDINES FOR CONTROLLING HELICOBACTER BACTERIA Compounds having the formula (I), in which R1, R2, R3, R4, R5, R6, R7, m, n and p have the meanings given in the description, are suitable for controlling helicobacter bacteria.
WO/1994/019321A1	INHIBITORS OF HIV REVERSE TRANSCRIPTASE Novel indole compounds inhibit HIV reverse transcriptase, and are useful in the prevention or treatment of infection by HIV and the treatment of AIDS, either as compounds, pharmaceutically acceptable salts, pharmaceutical composition ing...
WO/1994/019329A1	SUBSTITUTED CYCLIC CARBONYLS AND DERIVATIVES THEREOF USEFUL AS RETROVIRAL PROTEASE INHIBITORS This invention relates to substituted cyclic carbonyls and derivatives thereof useful as Human Immnunodeficiency Virus (HIV) protease inhibitors, to pharmaceutical compositions comprising such compounds, and to methods of using these com...
WO/1994/018174A1	SUBSTITUTED TETRAHYDROPYRIDAZINE CARBOXAMIDES The present invention pertains to new substituted tetrahydropyridazine carboxamides of general formula (I), in which R1 stands for hydrogen or alkyl, R2 stands for alkyl carbonyl or alkoxy carbonyl or R1 and R2 together with the nitrogen...
WO/1994/018177A1	ARYLAMINOSULPHONYL UREAS The invention relates to novel arylaminosulphonyl ureas of the general formula (I) in which R1 is possibly substituted alkyl with 2 to 10 carbon atoms, aryl or aralkyl, R2 is hydrogen, hydroxy, cyano, alkoxycarbonyl or possibly substitut...
WO/1994/018176A1	ARYLAMINOSULPHONYL UREAS The invention relates to novel arylaminosulphonyl ureas of the general formula (I) in which n represents the figures 1 or 2, R1 is possibly substituted alkyl, aryl or aralkyl, R2 is hydrogen, hydroxy, cyano, alkoxycarbonyl or possibly su...
WO/1994/014793A1	CYCLIC SULFONE CONTAINING RETROVIRAL PROTEASE INHIBITORS The present invention relates to cyclic sulfone moiety-containing hydroxyethylamine protease inhibitor compounds and pharmaceutical or method of use therefor, particularly as an inhibitor of HIV protease.
WO/1994/014767A1	PHENYL DERIVATIVES USEFUL AS TACHYKININ ANTAGONISTS Compounds of formula (I), or a salt or prodrug thereof are tachykinin antagonists.
WO/1994/014436A1	RETROVIRAL PROTEASE INHIBITING COMPOUNDS A retroviral protease inhibiting compound of formula (A) is disclosed.
WO/1994/014761A1	ARALKYLOXY- AND ARALKYLTHIO ALKOXIMINO DERIVATIVES AND THEIR USE AS FUNGICIDES A compound having general formula (I), wherein R1 and R2 are independently hydrogen, C1-4 alkyl, C1-4 haloalkyl, C2-4 alkenyl, C2-4 alkynyl, C3-6 cycloalkyl, aryl or aryl(C1-4)alkyl; R3 is hydrogen, C1-4 alkyl, C1-4 haloalkyl or C3-6 cyc...
WO/1994/014742A1	TRI-SUBSTITUTED PHENYL DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS Compounds of general formula (1) are described wherein Y is a halogen atom or a group -OR1, where R1 is an optionally substituted alkyl group; X is -O-, -S- or -N(R8)-, where R8 is a hydrogen atom or an alkyl group; R2 is an optionally s...
WO/1994/013712A1	MONOMER PRESENTING AT LEAST ONE ISOCYANATE FUNCTION AND AN INSATURATION, SYNTHESIS PROCESS AND (CO)POLYMERS DERIVED THEREFROM The monomer is characterized by the general formula (1) [(R1)(R2)C = C(R3)-CO-L-]q A(NCObloc)p wherein R1, R2 and R3 similar or different, represent a hydrogen or a group selected among the hydrocarbon chains having from 1 to 12 carbon a...
WO/1994/013645A1	NOVEL SELECTIVE AROMATASE INHIBITING COMPOUNDS New compounds of formula (I) wherein R1 is H, CH3, OCH3, NO2, NH2, CN, CF3, CHF2, CH2F or halogen, R2 is a heterocyclyl radical selected from 1-imidazolyl, triazolyl, tetrazolyl, pyrazolyl, pyrimidinyl, oxazolyl, thiazolyl, isoxazolyl an...
WO/1994/013652A1	HERBICIDES A compound of formula (I), where E is oxygen or sulphur; A is CR3 or N where R3 is hydrogen or hydrocarbyl; D completes a 5 or 6-membered non-aromatic heterocyclic ring which optionally contains additional heteroatoms selected from oxyge...
WO/1994/012181A1	FIBRINOGEN RECEPTOR ANTAGONISTS Novel fibrinogen receptor antagonists of the formula: X-Y-Z-Aryl-A-B are provided in which the claimed compounds exhibit fibrinogen receptor antagonist activity, inhibit platelet aggregation and are therefore useful in modulating thrombu...
WO/1994/012461A1	CATECHOL DIETHERS AS SELECTIVE PDEIV INHIBITORS This invention relates to 4-substituted catechol diether compounds which are selective inhibitors of phosphodiesterase (PDE) type IV. The compounds of the present invention are useful in inhibiting PDEIV and in the treatment of AIDS, ast...
WO/1994/011359A1	PROCESSES FOR PREPARING 2,4-OXAZOLIDINEDIONES Processes for preparing 2,4-oxazolidinediones having formula (I) wherein: R1 is phenyl optionally substituted with 1-2 halogen; or 4-phenoxy, 4-(1-phenethyloxy) or 4-benzyloxy each optionally substituted with R2 on the phenyl ring; and R...
WO/1994/011340A1	HYDRAZONE DERIVATIVE A compound representd by general formula (I), a salt thereof, and a pest control agent, wherein: X represents halogen, alkyl, alkoxy, cycloalkyloxy, alkylsulfonyloxy, alkylthio or alkylsulfonyl; R1 represents hydrogen or alkyl; R2 repres...
WO/1994/011278A1	CONTAINER FOR COLLECTING ORGANIC WASTE A container (1) is disclosed for collecting, composting or fermenting organic waste produced in households, small industries or the like. A venting hole (2) is arranged in the upper area of the collecting container and a biofilter (3) is...
WO/1994/011358A1	SULPHONYL UREA COMPOUNDS WITH A HERBICIDAL ACTION, METHOD OF PREPARING THEM AND THEIR USE Described are sulphonyl urea compounds of the general formula I in which R1 is a methyl or ethyl group; R2 is C1-C3 alkoxycarbonyl, a C1-C2 alkyl group with 1 to 5 fluorine atoms, methylsulphonyl, dimethylaminosulphonyl, thiomethyl, meth...
WO/1994/011364A1	PROCESS FOR PREPARING ENANTIOMERICALLY PURE 6-[(4-CHLOROPHENYL)(1H_-TRIAZOL-1,2,4-TRIAZOL-1-YL)METHYL]-1-METHYL-1H_-BENZOTRI AZOLE A process for preparing (+)-6-[(4-chlorophenyl)(1H_-1,2,4-triazol-1-yl)methyl]-1-met hyl-1H_-benzotriazole comprising the resolution of (U)-6-[(4-chlorophenyl-hydrazinomethyl)-1-methyl-1H_-benzotr iazole and converting the appropriate en...
WO/1994/011352A1	2-CYANO-SUBSTITUTED BENZIMIDAZOLES, THEIR PRODUCTION AND THEIR USE AS PESTICIDES The invention relates to the use of partly novel substituted benzimidazoles of general formula (I) where X1, X2, X3 and X4 are mutually independently hydrogen, halogen, cyano, nitro, possibly substituted alkyl, alkoxy, alkylthio, alkylsu...
WO/1994/010164A1	4-QUINOLINYL DERIVATIVES WITH ANTI-HELICOBACTER ACTIVITY The present invention is concerned with novel quinoline derivatives having anti-Helicobacter activity of formula (I), the pharmaceutically acceptable acid addition salts therof, the stereochemically isomeric forms thereof, the quaternize...
WO/1994/010154A1	NEW PHENYLSULPHONYL UREAS, THEIR PREPARATION AND THEIR USE AS HERBICIDES AND PLANT-GROWTH REGULATORS Described are compounds of the formula (I) in which R1 to R4, W, X, Y and Z are as defined in claim 1. Such compounds are suitable for use in the control of weeds in crops. Intermediates of the formulae (II) and (III) may be used to prep...
WO/1994/010142A1	NEW SUBSTITUTED AZETIDINONES AS ANTI-INFLAMMATORY AND ANTIDEGENERATIVE AGENTS Substituted azetidinones of general formula (I) which have been found to be potent elastase inhibitors and thereby useful anti-inflammatory and antidegenerative agents, wherein: R4 is (a) or (b) where Rx is carboxy C1-6alkyl, benzyloxyca...
WO/1994/010165A1	4-ARYLMETHYLOXYMETHYL PIPERIDINES AS TACHYKININ ANTAGONISTS Compounds of formula (I) wherein m is 2, 3 or 4; n is 0, 1 or 2 when m is 2 or 3, and n is 0 or 1 when m is 4; X represents O or S; R1 represents phenyl optionally substituted by 1, 2 or 3 groups selected from C1-6alkyl, C2-6alkenyl, C2-...
WO/1994/008973A1	AZOLE COMPOUND A compound represented by general formula (I), wherein R1 represents imidazolyl, triazolyl or tetrazolyl each of which may be substituted by methyl and/or ethyl. R2 represents naphthyl, phenanthryl or anthryl each of which may be substit...
WO/1994/008582A1	VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST A benzazepine compound represented by formulae (I) or (II) or a salt thereof, and a vasopressin antagonist or an oxytocin antagonist containing the above compound as the active ingredient.
WO/1994/008943A1	2-AMINO-1,3-PROPANEDIOL COMPOUND AND IMMUNOSUPPRESSANT A 2-amino-1,3-propanediol compound represented by general formula (I) or a pharmaceutically acceptable salt thereof, and an immunosuppressant containing the same as the active ingredient. In said formula R represents optionally substitut...
WO/1994/008972A1	OLIGOMERIC HETEROCYCLIC SALTS AND THEIR USE AS ANTIMICROBIAL AGENTS IN SWIMMING POOLS AND SPAS The use of oligomeric imidazolium, pyrazolium and triazolium salts of formula (I) as swimming pool sanitizers having improved compatibility with chlorine. Bisimidazolium salts are preferred.
WO/1994/008978A1	FUNGICIDAL SUBSTITUTED AZOLE DERIVATIVES Compounds having the structural formula (I), wherein R can be the same or different and is halogen, hydrogen, C1-C8 alkyl, C1-C8 haloalkyl, C3-C6 cycloalkyl, C7-C9 aralkyl, phenyl, nitro, C1-C6 alkoxy, C1-C6 alkylthio, C1-C6 alkylsulfiny...

Matches 1,201 - 1,250 out of 5,408	< 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 >