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Matches 301 - 350 out of 629

Document Document Title
JP4153057B2
Trehalose is oxidized to give oxidized trehalose which then is hydrolyzed to produce D-glucuronolactone which is thereafter recovered to realize high-yield and low-cost production of D-glucuronolactone.  
JP4097294B2
The present invention describes a method for treating neuropathic pain comprising administering to a mammal afflicted with such condition a therapeutically effective amount for treating such condition of a compound of formula (I), wherei...  
JP2007530700A
Compounds and methods useful in the control, treatment, and prevention of fungal activity, of the following formula: where R1-3 are independently H, alkyl, methyl, acyl, halogen, phenyl, R4 is H, alkyl, methyl, acyl, alkoxy, halogen, phe...  
JP3992510B2  
JP2007527520A
Methods are disclosed for providing a library of composite or novel composition samples on a support. The method involves depositing one or more components as concentration gradients on the surface of the support. The concentration gradi...  
JP3942414B2
To provide a new efficient synthesis method for industrially producing an L-type nucleic acid derivative as a medicine. A method by which the L-type nucleic acid derivative can industrially be produced from L-arabinose, one of few indust...  
JP2006232861A
To provide a novel efficient synthetic method for industrially producing an L-nucleic acid derivative as a medicine.Provided is the method industrially producing the L-nucleic acid derivative in a short process by using L-arabinose which...  
JP2006518759A
It is taught here that enkephalin peptides which are glycosylated with a disaccharide will be transported across the blood brain barrier and deliver analgesic effects superior to morphine when introduced into the bloodstream. Glycosylate...  
JP3789951B2
PURPOSE: To obtain a new compound capable of producing hydantocidin in high yield without forming stereoisomers. CONSTITUTION: This sugar derivative is a compound of formula I [R1 and R2 each is H or together form a (substituted) alkylid...  
JP2006514071A
The invention relates to novel pharmaceutically acceptable salts of anticonvulsant derivatives, processes for preparation of and pharmaceutical compositions containing said salts, useful in the treatment of epilepsy.  
JP2006052182A
To provide a method for producing a fluorinated purine nucleoside derivative, by which the 3-position (preferably the α-position) is economically and efficiently fluorinated and which is suitable for industrial production.This method fo...  
JP2006502103A
The invention relates to a novel palatinose condensation product which is obtained by condensing the disaccharide palatinose in a molten mass of palatinose, water and an organic acid.  
JP3725233B2
To obtain a trehalose derivative excellent in surface-active ability and safety to skin and useful as a surfactant, etc., capable of using for cosmetics, medicines, foods, etc., by reacting trehalose with an acetal compound in the presen...  
JP2005536493A
This invention relates to processes for production of alkylamino glucosaminide phosphate compounds, and of disaccharide compounds, including various novel intermediates and intermediate processes. In one aspect, glycosyl halides are prod...  
JP2005289964A
To provide an efficient production method of a 2-deoxy-L-ribose compound and its protection compound.This production method comprises reacting an aldehyde compound represented by formula (1) (wherein R1 and R2 are each independently or i...  
JP3706875B2
To provide tea leaves with reduced caffeine content, capable of being taken by a large amount for a long time as an antiallergic beverage or food. A method for producing tea leaves is provided by immersing any of raw leaves of "Benifuuki...  
JP2005530808A
This invention relates to a new pharmaceutically useful compound which is a stoichiometrically 1:1 adduct of tramadol hydrochloride and topiramate, to the manufacture and use thereof.  
JP2005526852A
The present invention is directed to novel compounds of the formula (I) wherein X, R1, R2, R3, R4, R5 and R6 are as described in the specification, processes for the preparation of and pharmaceutical compositions comprising said derivati...  
JP3662954B2
PURPOSE: To obtain the subject compound, useful for a raw material, etc., for liquid crystals, medicines, agrochemicals, etc., by optically resolving a recemic 1-benzyloxy-6,6,6-trifluoro-4-hexyn-3-ol, then carrying out the reduction of ...  
JPWO2003072587A1
本出願には、システイン若しくは/およびシ ステイニルグリシンまたはシスチンと還元糖 とを水性溶媒中に加熱下に保持することを特 徴とする不揮発性チアゾリジン化合物の...  
JP2005514352A
The present invention is directed to a method for treating autoimmune diseases comprising administering a therapeutically effective amount of a compound of the following formula (I) wherein X, R1, R2, R3, R4, R5 and R6 are as herein defi...  
JP3621097B2
The present invention relates to a method of preparing BCH-189 and various analogues of BCH-189 from inexpensive precursors with the option of introducing functionality as needed. This synthetic route allows the stereoselective preparati...  
JP2005503358A
The present invention includes compounds and compositions of beta-halonucleosides, as well as methods to treat HIV, HBV or abnormal cellular proliferation comprising administering said compounds or compositions.  
JP3602050B2
A composition comprises 12,13-(Pyranosyl)-indolo(2,3-a)pyrrolo(3,4-c)carbazole and 12,13-(pyranosyl)-furo(3,4-c)indolo(2,3-a)carbazole derivatives (I), or their isomers, salts with acids or bases, are new A composition comprises 12,13-(P...  
JP2004262911A
To provide a method for producing effectively an optically active α-aminoketone.A method for producing an optically active α-aminoketone shown by general formula (2) comprises allowing a new chiral alkoxide originating from glucose, wh...  
JP2004523478A
The present invention relates to novel N12, N13-bridged sugar derivatives of indolylopyrrolocarbazoles and pharmaceutical formulations thereof which exhibit topoisomerase-I activity and are useful in inhibiting the proliferation of tumor...  
JP2004518803A
Avilamycin derivatives, gene technology biosynthesis processes for their production, medications containing these compounds, as well as the use of these compounds for the production of a active agent against infectious diseases, as well ...  
JP2004175792A
To provide a method for simply producing a 2,2'-anhydro-1-(β-D-arabinofuranosyl)uracil compound at a low cost.This method for producing the 2,2'-anhydro-1-(β-D-arabinofuranosyl)uracil compound comprises heating a 3',5'-O-sulfinylxylour...  
JP2004517932A
The present invention provides stable compounds prepared from boronic acid and lyophilized compounds thereof of formula (1) in which Z 1 and Z 2 are moieties derived from sugar. The invention also provides methods for preparing such comp...  
JP2004123605A
To provide a method for highly selectively, efficiently and safely advancing the fluorination reaction of a desired substrate.This fluorination method comprises reacting a specific fluorine compound such as N, N-diethyl-α, α-difluoro-(...  
JP3516959B2
Methods and compositions are provided which increase the cellular uptake of bioactive materials by covalently bonding such compounds to carbohydrate moieties through chemical linkers using other than glycosidic bonds. Numerous carbohydra...  
JP2003530300A
Anticonvulsant derivatives useful in maintaining weight loss.  
JP2003527324A
Heterocyclic aromatic amides (HAA) according to Formula (I) wherein X1-X4, M, Z, and A are herein defined. The invention also encompasses hydrates, salts and complexes thereof. These compounds are useful as antifungal agents.  
JP3430318B2
PURPOSE: To provide halistatin 1 which is useful as a material for anticancer drugs. CONSTITUTION: Halistatin 1 is shown by the formula. This compound is obtained from the sponge Phkellia-carteri gathered in the west Indian Ocean by extr...  
JP3430317B2
PURPOSE: To provide halistatin 2 which exerts, as an anti-tumor agent, a particularly excellent activity against leukemia, small cell carcinoma of lung, large bowel cancer, CNS cancer and melanoma. CONSTITUTION: The halistatin 2 is shown...  
JP2003176250A
To provide a method of synthesizing phosphine oxide being a synthon for ring A used for preparing 19-nor-vitamin D compound and provide a new synthetic intermediate that is formed on the way of the synthetic route.In this new synthetic p...  
JP3411280B2
A method for vacuum distillation includes separation of a liquid product delivered to a reservoir under vacuum into a vapour-gaseous phase and at least one liquid fraction, withdrawal of the vapour-gaseous phase from the reservoir using ...  
JP3403218B2
PURPOSE: To provide a new compound useful as an antiliphemic and for treating liver disorders with cholestasis with no side-effects, which has activity to decrease the cholesterol level in the serum and has high affinity for transport sy...  
JP2003055394A
To provide a synthetic compound which is useful for obtaining an oligo saccharide specifically bound to a target nucleic acid in the specific sequence of a gene, and to enable the enhancement in the effect of an anti-gene method. This di...  
JP2003505465A
Anticonvulsant compounds of the general formula I:where X, R1, R2, R3, R4, R5, and R6 are as herein defined; are useful in treating acute ischemia-induced neurodegeneration, such as occurs during and after stroke, head trauma, spinal inj...  
JP2003502325A
The invention relates to a method for the enantiomer separation of cis-8-benzyl-7,9-dioxo-2,8-diazabicy-clo[4.3.0]nonane (also described below as cis-6-benzyl-5,7-dioxooctahydropyrrolo[3,4-b]pyridine or dioxopyrrolopiperidine). The inven...  
JP2002544135A
Synthetic methods for convenient large scale preparation of D-erythro sphingosines and ceramides of high isomeric purity are described.  
JP2002543214A
Provided are L-ribo bicyclic nucleotide compounds as well as syntheses of such compounds. The nucleoside compounds of the invention are useful in forming oligonucleotides that can produce nucleobase specific duplexes with complementary s...  
JP3356324B2
Compounds of the general formula (I): wherein R1, R2, R3, R4, R5, R6, n and p are as herein defined; exhibit anticonvulsant activity and are thus useful in the treatment of conditions such as epilepsy. Compounds of this class are also us...  
JP2002537264A
The present invention relates to benzaldehyde derivatives which are useful as anticancer agents. Some of the compounds of this invention are novel per se.  
JP2002537263A
The present invention relates to benzaldehyde derivatives which are useful as anticancer agents. Some of the compounds of this invention are novel per se.  
JP2002536328A
Anticonvulsant derivatives useful in treating autism.  
JP2002535270A
Anticonvulsant derivatives useful in treating cluster headaches are disclosed.  
JP2002534529A
The present application relates to a group of novel substituted pentose and hexose monosaccharide derivatives, not previously disclosed, which exhibit potent anti-cell adhesion and anti-inflammatory activities. Methods of preparation, ph...  
JP2002534530A
This invention relates generally to compounds and processes for synthesizing derivatives of 2-3-O-isopropylidene-alpha-L-xylo-2-hexulofuranosonic acid. The compounds of this invention are useful, inter-alia, for the inhibition and preven...  

Matches 301 - 350 out of 629