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WO/1996/021354A1 |
Pesticidal as a pesticide against whitefly, Lepidoptera and certain fungi is provided of compound of general formula (I) or a salt thereof is provided, in which n represents an integer from 0 to 4; m represents an integer 0 or 1; each R ...
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WO/1996/021638A1 |
A compound of formula (I), or a salt thereof, or a solvate thereof, wherein: R1 is an alkyl group or a substituted or unsubstituted phenyl group; R2 and R3 each independently represent hydrogen or alkyl; and either: RA represents T1 wher...
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WO/1996/020914A1 |
Tricyclic retinoids having activity for retinoic acid receptors and/or retinoid X receptors are provided. Also provided are pharmaceutical compositions incorporating such tricyclic retinoid compounds and methods for their therapeutic use.
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WO/1996/019988A1 |
The present invention relates to novel 4,4-(disubstituted)cyclohexan-1-ols monomers and related compounds, pharmaceutical compositions containing these compounds, and their use in treating allergic and inflammatory diseases and for inhib...
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WO/1996/020158A1 |
This invention relates to derivatives of 3,3-(disubstituted)cyclohexan-1-one monomers and related compounds which are useful for treating allergic and inflammatory diseases.
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WO/1996/019288A1 |
Porous microcomposites have been prepared from perfluorinated ion-exchange polymer and metal oxides such as silica using the sol-gel process. Such microcomposites possess high surface area and are useful as catalysts for olefin isomeriza...
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WO/1996/018607A1 |
A compound represented by general formula (1) or possible stereoisomers and optical isomers thereof, and medicinally acceptable salts of these compounds, wherein R1 represents SR6 or NHR7; R6 represents C1-C6 alkyl, etc.; R7 represents h...
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WO/1996/018605A1 |
This invention relates to novel acyloxyisopropyl carbamates as bioreversible prodrug moieties for amino drugs and to methods of synthesizing these compounds.
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WO/1996/018608A1 |
A compound represented by general formula (1),zor possible stereoisomers and optical isomers thereof, and medicinally acceptable salts of these, (wherein R1 represents SR6 or NR7R8; R6 represents C1-C6 alkyl, etc.; R7 represents hydrogen...
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WO/1996/016030A1 |
Iminooxymethylene anilides have the formula (I), in which the substituents and indices have the following meanings: R stands for hydrogen, optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, cycloalkinyl, alkylcarbo...
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WO/1996/015084A1 |
A process for producing a halogenated organic compound by the addition reaction between an organic compound having an aliphatic carbon-carbon unsaturation and a hydrogen halide, wherein the reaction is catalyzed by an organic compound ha...
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WO/1996/015090A1 |
A nonsolvent process of synthesizing bis(2,2-dinitropropyl)formal (BDNPF) is disclosed. In the process, 2,2-dinitropropanol (DNPOH) is reacted at low temperature with a formaldehyde source in the presence of a protic acid catalyst, such ...
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WO/1996/015096A1 |
Inhibitors for matrix metalloproteases, pharmaceutical compositions containing them, and a process for using them to treat a variety of physiological conditions. The compounds of the invention have the generalized formula (T)xA-B-D-E-G, ...
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WO/1996/015092A1 |
Fluorine-containing liquid crystal compounds comprise a fluorocarbon terminal portion having at least one catenary ether oxygen and a hydrocarbon terminal portion, the terminal portions being connected by a central core. The compounds ha...
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WO/1996/015091A1 |
A nonsolvent process of synthesizing bis(2,2-dinitropropyl)acetal (BDNPA) is disclosed. In the process, 2,2-dinitropropanol (DNPOH) is reacted at low temperature with an acetaldehyde source in the presence of an acid catalyst, such as a ...
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WO/1996/014285A1 |
A substituted bicycloheptanedione derivative represented by general formula [I], its salts, and a herbicide containing the same as the active ingredient, wherein R represents C1-C4 alkyl; R1 represents hydrogen, C1-C10 alkyl, C2-C4 alken...
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WO/1996/014298A1 |
Disclosed are substituted phthalimido-cinnamic acid derivatives of formula (I), wherein R1 is H, C1-C4-alkyl; R2 is H, halogen; R3 is CN, NO2, halogen, C1-C6-alkyl, C1-C6-alkyl halide, C1-C6-alkoxy, C1-C6-alkoxy halide; R4 is H, CN, NO2,...
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WO/1996/013569A1 |
Disclosed is a single phase mixture of about 1 to about 99 wt% of a compound having general formula (I) where "n" is 1 or 2 and about 0.1 to about 99 wt% of a liquid which can be a perfluoro aliphatic alkane from C5 to C8, a perfluoro cy...
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WO/1996/013491A1 |
Compounds having the formula (I): R1R2C(OR3)-Ar1-X-Ar2-C(Ar3)=CHCO2H are inhibitors of leukotriene biosynthesis. These compounds are useful as anti-asthmatic, anti-allergic, anti-inflammatory, and cytoprotective agents. They are also use...
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WO/1996/012725A1 |
The description relates to quinoxalindione derivatives (I) and their production and use in medicaments.
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WO/1996/011902A1 |
The present invention relates to compounds of formula (I), wherein: A, B and D are various ring systems as defined in the description, R1 is one of a variety of groups as defined in the description, R3 is hydrogen or C1-4 alkyl and Z is ...
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WO/1996/010561A1 |
2-aroylcyclohexandiones have general formula (I), in which X, Y stand for O or S; Ar stands for phenyl or heteroaryl with 1 to 4 substituents; or two adjacent carbon atoms of the phenyl or heteroaryl ring may also be bridged by a chain; ...
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WO/1996/010004A1 |
A process for the purification of 2,6-diisopropylphenol (Propofol) by transformation of the crude Propofol into its ester with a carboxylic or sulphonic acid, crystallization and hydrolysis, is described.
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WO/1996/010010A1 |
A method for preparing a compound of formula (I), wherein R1 and R2, which are the same or different, are a hydrogen atom or an alkyl or alkoxy radical, or R1 and R2, taken together with the carbon atom to which they are attached, form a...
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WO/1996/009275A1 |
The present invention concerns novel fullerene derivatives of the formula (I) in which the symbols and indices mean: F - a fullerene radical of the formula C20+2m, where m = 2 to 100; R1 - an aryl radical which may be substituted by 1 to...
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WO/1996/009274A1 |
The invention provides a method for the preparation of 3,4-dihydroxy-5-nitrobenzaldehyde by reacting 3-ethoxy-4-hydroxy-5-nitrobenzaldehyde with a reagent comprising zinc chloride, water and hydrogen chloride.
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WO/1996/006822A1 |
The present invention relates to compounds of formula (I) wherein: A is an optionally substituted ring system as defined herein; B is an optionally substituted 5- or 6-membered heteroaryl ring system or optionally substituted phenyl; D i...
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WO/1996/003367A1 |
The invention concerns reaction products of polyisobutylenes having an average polymerisation degree P of 10 to 100 and a proportion E of 60 to 90 % of double bonds which can be reacted with maleic acid anhydride, E corresponding to 100 ...
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WO/1996/003356A1 |
A method of iodinating and/or brominating and/or chlorinating an aromatic compound which comprises the steps of reacting an iodinating agent and/or brominating agent and/or chlorinating agent with the aromatic compound in the presence of...
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WO/1996/002515A1 |
The disclosure herein relates to the title compounds of formula (I) and salts and esters thereof, wherein X is halogen, C1-6 polyhaloalkyl, C6-10 aryloxy, C1-6 alkoxy or alkylsulfonyl, C4-10 tert-alkyl, NO2 or CN; n is 0-4 and Z is an (u...
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WO/1996/002493A1 |
A method useful for the synthesis of a meta-substituted nitrogen derivative, comprising the step of deaminating an ortho- and/or para-substituted nitroaniline of the aniline function. The method is useful for organic synthesis.
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WO/1996/002491A1 |
Photoreactive compounds are synthesized from 2,5- or 2,6-dinitrobenzyl groups. Also disclosed are methods of synthesizing reactive monomers containing 2,5- or 2,6-dinitrobenzyl groups.
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WO/1996/001798A1 |
The present invention relates to novel 2-aryl-3-hydroxy-cyclopenet-2-en-1-one derivatives of formula (I) in which X is halogen, nitro, cyano, alkyl, alkoxy, alkenyloxy, alkylthio, alkyl sulphinyl, alkyl sulphonyl, halogen alkyl or haloge...
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WO/1996/001258A1 |
The invention concerns 2-[1',2',4'-triazol-3'-yloxymethylene]-anilides of the formula (I) in which the subscript and substituents are as follows: n stands for 0, 1, 2, 3, or 4; X stands for a direct bond, oxygen or NRa, Ra being hydrogen...
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WO/1996/000378A1 |
Novel compounds are provided which are useful as photocleavable linking groups in solid phase synthesis. Compositions incorporatinf these linking groups and methods for their use are also described.
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WO/1995/035284A1 |
Compounds of general formula (1) are described wherein =W- is (1) =C(Y)- where Y is a halogen atom, or an alkyl or -XRa group where X is -O-, -S(O)m-[where m is zero or an integer of value 1 or 2], or -N(Rb)- where Rb is a hydrogen atom ...
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WO/1995/031429A1 |
This invention relates to agents and conjugates that can be used to detect and isolate target components from complex mixtures such as nucleic acids from biological samples, cells from bodily fluids, and nascent proteins from translation...
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WO/1995/030642A1 |
Combinatorial libraries are disclosed which are represented by the Formula (I): (T'-L)q- S -C(O)-L'-II' wherein S is a solid support; T'-L- is an identifier residue; and -L'-II' is a ligand/linker residue. These libraries contain dihydro...
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WO/1995/030641A1 |
New compounds and their compositions having anti-inflammatory, analgesic and anti-thrombotic activities, of the general formula: A-X1-NO2 or their salts, wherein: A is R(COXu)t, wherein t is zero or 1 and u is zero or 1; and X is O, NH o...
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WO/1995/029886A1 |
The present invention concerns processes for preparing aromatic, bromine-containing compounds, novel bromine-containing compounds and their use as intermediate products in the synthesis of active agents. Processes according to the invent...
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WO/1995/028640A1 |
Encoded combinatorial chemistry is provided, where sequential synthetic schemes are recorded using organic molecules, which define choice of reactant, and stage, as the same or different bit of information. Various products can be produc...
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WO/1995/025710A1 |
A triphenylene such as hexa-'beta'-substituted hexyloxytriphenylene is 'alpha'-substituted by an electrophile in mixed polar cosolvents according to the reaction scheme (a).
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WO/1995/024897A1 |
2-Chloro-5-nitrobenzoic acid and various other chloro and nitro substitute benzoic acid derivatives are disclosed for administration in tablet or injectable solution form for the prophylaxis and therapy of neoplasm or viral infection. Th...
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WO/1995/025085A1 |
4, 6-Dinitroresorcinol is prepared by reacting resorcinol with concentrated nitric acid that is substantially free of suboxides of nitric acid. It has been found that greater than 60 percent yields of the desired product can be obtained ...
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WO/1995/024454A1 |
The invention concerns mixtures of liquid-crystalline compounds containing at least two different substances of general formula (I) in which the radicals Z1, Z2, independently of one another, mean a polymerisable group, Y1, Y2, independe...
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WO/1995/024397A1 |
A compound having the formula (I), a physiologically tolerable salt of the compound having the formula (I) and/or a stereoisomeric form of the compound having the formula (I), in which one residue R1 or R2 stands for the formula (II), ar...
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WO/1995/024186A1 |
Combinatorial libraries are disclosed which are represented by the formula (I): (T'-L)q- S -C(O)-L'-II' wherein: S is a solid support; T'-L- is an identifier residue; and -L'-II' is a ligand/linker residue. These libraries contain aryl s...
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WO/1995/021610A1 |
Products having formula (I) wherein R2 is (C1-C4)-alkyl, (C1-C4)-acyl, CF3, Cl, Br or I; R3 is H, (C1-C4)-alkyl, (C1-C4)-acyl, (C1-C4)-alcoxyl, CF3, F, Cl, Br, phenyl, OH, SH, NH2 or amino mono- or bisubstituted by (C1-C3)-alkyl; R4 is (...
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WO/1995/021153A1 |
Phenyl acetic acid derivatives of formula (I) in which the components and index have the following meanings: X is NOCH3, CHOCH3 CHCH3 and CHCH2CH3; R1 is hydrogen and alkyl; R2 is cyano, nitro, trifluoro methyl, halogen, alkyl and alkoxy...
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WO/1995/021149A1 |
A cyclooctadiene derivative represented by general formula (I), and an agrohorticultural bactericide, antimold and antithrombocytic agent each containing the derivative (I) (i) or (ii), wherein A1 to A4 represent each COOR5 (R5 being H, ...
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