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JPH02138245A |
NEW MATERIAL: A compounds of formula I [R1 is a 1-4C alkyl, a 2-3C alkenyl or alkynyl, a 3-4C haloalkenyl having 1-3 halogen, etc.; R2 is a 1-4C alkyl; R3 is formula II (X is O or S; R4 and R5 are each a 1-4C alkyl, commonly an alkylene)...
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JPH02501388A |
PCT No. PCT/CH88/00163 Sec. 371 Date May 19, 1989 Sec. 102(e) Date May 19, 1989 PCT Filed Sep. 19, 1988 PCT Pub. No. WO89/02891 PCT Pub. Date Apr. 6, 1989.The invention is concerned with novel compounds of the formula I wherein R1, R2, R...
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JPH02124859A |
NEW MATERIAL: A compound of formula I [wherein the symbol CYCLE together with the C atoms bonded to the semicircle is a four- or seven-membered carbocyclic or heterocyclic ring having an ethylenic or aromatic unsaturation between the two...
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JPH02501140A |
Novel renin-inhibitory peptides of the formula X-A6-B7-C8-D9-E10-F11, containing C-terminus truncated epoxy or azido or cyano groups or containing a position 10-11 diol and a position 11-12 retro bond. The present invention further provi...
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JPH0288553A |
NEW MATERIAL: (E)-N-{1(S)-methyl-3-[3-(4-fluorophenoxy)phenyl]prop-2-en-l-
yl}acetohydroxamic acid and its salt. USE: This new material is useful as an inhibitor of lipoxygenase and cyclo- oxygenase and also useful for treating and prev...
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JPH0285241A |
PURPOSE: To provide a compd. used for preparing a medicine which has a specified compd. contg. a new compd. as an active ingredient and exhibits excellent bronchodilator activity and can be administered through various paths such as oral...
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JPH0242052A |
NEW MATERIAL: A compd. represented by formula I [wherein A1 to A3 are carbamoyl having the partial formula; -CO-NH-AlK-CO-O-R11 (wherein Ra1 is a 1-4C alkyl or 2-4C alkenyl, AlK is a non-substituted or hydroxy or 1-4C alkanoyloxy), H or ...
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JPH0236163A |
NEW MATERIAL: A compd. represented by formula I [wherein RCO is an acyl residue of a non-steroidal anti-inflammatory drug, R1 is H, an alkyl or acyl, R2 is H, an alkyl, cycloalkyl, aryl, arylalkyl or heteroaryl and an acyl residue is a g...
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JPH0236164A |
PURPOSE: To obtain the subject compound for herbicides by nitrating a readily available novel compound, such as O-methoxycarbonylmethyl-3-(2-chloro-4- trifluoromethylphenoxy)benzohydroximate. CONSTITUTION: A novel compound expressed by f...
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JPH0217147A |
NEW MATERIAL: Compounds given by formula I [Y is OR1 (R1 is H or 1-4C alkyl), Cl, CH3, formula II (R2 is 1-4C alkyl), formula III (R3=R2) or formula IV; X is F, Cl, or Br; when Y is OH, X ≠ Br, when Y is CH3, X ≠ F is excluded; only ...
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JPH026423A |
NEW MATERIAL: A compd. represented by formula I [wherein R1 is H, a halogen, CN or CF3, R2, R4 and R5 are H or a halogen, R3 is a halogen, CN, CF3, trifluoromethoxy or trifluoromethylsulfonyl, X is a halogen, Y is a halogen, CN, azido, t...
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JPH026452A |
NEW MATERIAL: A compound of formula I [wherein A is formula II or the like; R1 is H, CH3, CH2-CH3 or the luke; R2 is H, CH3, C6H5 or the like; Z is H, C(CH3)3 or the liked; m is 0 or 1; and n is 0-3]. EXAMPLE: cis-2-[[N-(hydroxyamino)-2 ...
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JPH021441A |
NEW MATERIAL: Compd. of formula I [wherein X is O, S and NOR1 (wherein R1 is H, an alkyl, an alkenyl, an acyl, etc.); R is H, a halogen, CN, SCN, NO2, CN, an alkyl, a phenyl, etc.; R2 is H, an alkyl or S-CCl3; R3 and R5 are each NO2, a h...
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JPH02733A |
NEW MATERIAL: Compounds of formula I [X is halogen; Y is NR2R3, formula II (W is O, S; Z is O, S, NR1; n is 1-4; R2, R3 are each alkyl, alkenyl, phenyl, etc.; R4 is R1; R5 is H, alkyl, alkenyl, cycloalkyl, phenyl, etc.); R1 is H, alkyl, ...
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JPH021434A |
NEW MATERIAL: Compounds of formula I (R1 is formula II, formula III, NH-R2, etc.; R2 is H, amino, OC-Y, -P-phenyl-CH-Y, (substituted)alkyl, cycloalkyl, aryl, etc.; Y is EDTA, DTPA, DOTA, HETA, TRITA, TETA; M is a metal ion) or their salt...
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JPH021442A |
NEW MATERIAL: Compd. of formula I [wherein R1 is H, F or Cl; R2 is H, a (substd.) alkyl, an alkynyl, a cycloalkyl or a (substd.) phenyl; R3 is H, an alkyl, OR4 (wherein R4 is H, an alkyl, a phenyl, a naphthyl, etc.); R2 and R3 form toget...
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JPH01272553A |
NEW MATERIAL:A compound expressed by formula I (R1 is H, lower alkyl or aryl) or salt thereof. EXAMPLE: Disodium 2-hydroxy-2-(hydroxycarbamoyl)-3-methylglutarate. USE: An antimicrobial agent and carbapenem based antibiotic substance capa...
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JPH01246251A |
NEW MATERIAL:A compound shown by formula I (Z is CX or N; X is H or halogen: R1 and R2 are lower alkyl). EXAMPLE: Methyl O-methoxycarbonylmethyl-3-(2-chloro-4-trifluoromethyl-3-(2- chloro-4-trifluoromethylpheooxy)benzohydroximate. USE: A...
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JPH01246250A |
NEW MATERIAL:A compound shown by formula l (Z is CX or N; X is H or halogen ; R is lower alkyl). EXAMPLE: Methyl 3-(2-chloro-4-trifluoromethylphenoxy)benzohydroximate. USE: A synthetic intermediate of herbicides and capable of introducin...
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JPH01233203A |
PURPOSE: To provide a herbicide composition composed of a 2-nitro-5-(substituted phenoxy)benzohydroximic acid derivative and N-phosphonomethylglycine, etc., and exhibiting high herbicidal effect especially by foliar treatment. CONSTITUTI...
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JPH01226865A |
NEW MATERIAL:A compound of formula I [R1 is lower alkyl; R2 is H or lower alkyl; R is (substituted) phenyl]. EXAMPLE: Methyl O-phenoxycarbonylmethyl-5-(2-chloro-4-trifluoromethylphenoxy
)- 2-nitrobenzohydroximate. USE: A herbicide. The c...
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JPH01226864A |
NEW MATERIAL:A compound of formula I (R1 is lower alkoxyalkyl or lower alkylthioalkyl; R and R2 are H or lower alkyl). EXAMPLE: Ethoxymethyl O-methoxycarbonylmethyl-5- (2-chloro-4-trifluoro- methylphexy)-2-nitrobenzohydroximate. USE: A h...
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JPH01216905A |
PURPOSE: To obtain a herbicide composition effective against wide variety of weeds, especially for the weeding of orchard, at a low rate of application without causing the problem of acute toxicity, by using a novel benzohydroximic acid ...
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JPH01216961A |
PURPOSE: To provide the subject preparation useful as a preventing and treating agent for ischemic circulatory diseases, organ inflammation, vulgaris psoriasis, arterial sclerosis, etc., and having low toxicity and a little adverse effec...
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JPH0134980B2 |
Phenylacetic acid derivatives of the formula wherein n is an integer of 2 to 5; R1 is hydrogen, halogen, trifluoromethyl, nitro or amino; R2 and R3 each independently is hydrogen or lower alkyl; or together form an ethylene group; X1 rep...
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JPH01157961A |
NEW MATERIAL: A compd. of formula I {where R1 is H, halogen, CN or CF; R2 is H or halogen; R3 is halogen, CF3, OCF3, SCF3, etc.; R4 is R2; X is N or CR5 (R5 is R2); A is optionally branched alkanediyl; and Z is CN or CO-Y [Y is halogen, ...
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JPH01153658A |
NEW MATERIAL: A compd. of the formula I (wherein each of X and Y is NR, O, S, the formula II or a single bond; with the proviso that at least one of X and Y is not a single bond; R is H or lower alkyl; (g) is 1 or 2; Z is aryl, aralkyl o...
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JPH01151546A |
Compounds of the formula (I): wherein: X = O, S, or NOH; R<1> is H or CH3; n = 1, 2, or 3; R<2>, R<3>, and R<4> are as defined in one of the following paragraphs a) R<2> and R<3> are independently Cl or Br, and R<4> is H; b) R<2>, R<3>, ...
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JPH01143856A |
NEW MATERIAL: A compd. of formula I [X is CR4, N; Y is formula II (R4 is H, a lower alkyl), O, S, NR4, etc.; Z is (CH2)nO ((n) is 0 to 5), (CH2)nS, C≡C, etc.; R1 is formula III (R5 is a lower alkyl, a monofluorolower alkyl, etc.), etc....
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JPH01135742A |
(57) [Abstract] Since this gazette is application data in front of an electronic application, the data of an abstract is not recorded.
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JPH01113334A |
NEW MATERIAL: A compd. expressed by formula I [wherein R1 is halogen, CN or CF3; R2 is H or halogen; R3 is halogen, CF3, OCF3, SCF3 or trifluoromethylsulfonyl; R4 is H or halogen; X is N or CR5 (R5 is R2); A is alkane-diyl which may be a...
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JPH01113331A |
NEW MATERIAL: A compd. expressed by formula I, (wherein R1 is H, halogen, cyano or CF3; R2, R4 and R5 are each H or halogen; R3 is halogen, cyano, CF3, OCF3; Z is halogen, OH, amino, alkylamino, alkenylamino, alkynylamino, arylamino, ara...
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JPS6466147A |
PURPOSE: To simply obtain the titled compound in high yield, by reacting a reaction product of an aromatic carboxylic acid derivative and hydroxylamine with a halogenoacetic acid in the presence of a metal hydroxide or metal carbonate an...
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JPS6445344A |
NEW MATERIAL: Compounds represented by the formula I (wherein: (q) is 1; (k) is 0; (p) is 1; Ar is a phenyl group optionally substituted by a 1-4C alkyl group or a halogen; L is -O-; Ar' is a 1,3- or 1,4-phenylene group; Y is (E)-CH= CH-...
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JPS6419047A |
NEW MATERIAL:A compound expressed by formula I (R1 is H, lower alkyl or aryl) or salt thereof. EXAMPLE: Diethyl 2-benzoyloxy-2-ethoxycarbonyl-3-methyl-glutarate. USE: A dehydropeptidase I inhibitor administered to humans or animals requi...
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JPS6413059A |
NEW MATERIAL:A compound expressed by formula I (X is -COCH3 or benzyl; R is benzyloxy). EXAMPLE: (R)-N-Benzyloxy-4-acetoxy-3-hydroxy-butanamide. USE: A synthetic intermediate for optically active mono-β-latam rings. The above- mentioned...
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JPS6365138B2 |
A silver halide photographic light-sensitive material containing a diffusion resistant coupler, a light-sensitive silver halide and at least one compound represented by the following general formula (I) in the same layer or different lay...
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JPS6358820B2 |
The present invention relates as new industrial products to 4-phenoxy-3-butyramidoxime derivatives, characterized in that they are selected from the group consisting of 4-(allylphenoxy)-3-hydroxy-butyramidoximes of formula: (I) and addit...
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JPS63264442A |
Compounds of the formulae wherein n=6-11, M is hydrogen or a pharmaceutically acceptable cation, R is hydrogen or C1-C6 alkyl optionally substituted by a carboxyl group and Xa, Xb and Xc each independently represent hydrogen or a variety...
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JPS63258449A |
The compounds correspond to the general formula …… in which… -W denotes a residue of an amino acid chosen from valine, lysine, norleucine and methionine, and… -Z denotes an amino or alkylamino radical in which the alkyl part, whi...
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JPS63233950A |
NEW MATERIAL:A compound shown by formula I [R1 is hydroxyalkyl which may be protected; R2 is alkyl; R3 is R1, H or alkyltrisubstituted silyl; R4 is (substituted)OH or (substituted)amino or a salt thereof. EXAMPLE: 5-Benzyloxy-2-[1-tertia...
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JPS63225340A |
Compounds of the formula: where R1 is amino or methyl; R2 is C1-C2 alkyl; R3 is one or more substituents selected from hydrogen, halogen or trihalomethyl; R4 is one or more substituents selected from hydrogen, halogen, trihalomethyl, C1 ...
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JPS63215605A |
PURPOSE: To obtain a herbicide having wide herbicidal spectrum with a small application amount, showing excellent herbicidal selectivity even application to culture crops such as rice plant after germination, containing a specific (subst...
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JPS63183546A |
A new inclusion complex of ibuproxam with beta-cyclodextrin is described, which is prepared by adding ibuproxam to a boiling aqueous solution of beta-cyclodextrin, stirring the reaction mixture at the boiling temperature, cooling to a te...
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JPS63166856A |
NEW MATERIAL:The 2-nitro-5-(substituted phenoxy)benzohydroximic acid derivative of formula I [R1 is lower alkyl; R2 is H or lower alkyl; R is (substituted) alkenyl or (substituted)alkynyl]. EXAMPLE: Methyl O-allyloxycarbonylmethyl 5-(2-c...
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JPS63165359A |
NEW MATERIAL:A compound shown by formula I [X1 is halogen; X2 is H or halogen; X3 is halogen or trifluoromethyl; R1 and R2 are (i) lower alkyl, lower alkynyl, etc., or (ii) lower alkoxycarbonylalkyl, alkylcarbonyl, arylcarbonyl, etc., an...
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JPS6328060B2 |
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JPS63135360A |
NEW MATERIAL:The compound of formula I (X is halogen, lower alkyl, lower alkoxy, halo-lower alkyl or nitro; n is 0W2; R1 is lower alkyl, lower alkenyl, lower alkynyl or lower alkylthio-lower alkyl). EXAMPLE: Allyl phenylacetohydroxamate....
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JPS63130566A |
NEW MATERIAL:A compound expressed by formula I [A is formula II (X is halogen, CF3, lower alkyl, etc.; n is 0 or 1), etc.; R is H or lower alkyl; R1 and R2 are H, halogen or lower alkyl; R3 is H or tetrahydropyranyl; R4 is H, azide, etc....
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JPS6323987B2 |
The invention provides novel anti- atherosclerotic compounds of the type where A is the residue of a long chain, unsaturated fatty acid or cyclopropano analogues thereof; the -CO-N< moiety forms an amide or hydrazide group or the N atom ...
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