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JPH05239010A |
PURPOSE: To produce a 1.5-diaryl-3-formazancarbonitrile compd. useful as a treating agent or a systemic protective agent of domestic animals and fishes which are risked or liable to be risked by a parasite. CONSTITUTION: A compd. express...
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JPH05230009A |
PURPOSE: To provide a new amidine derivative having excellent fibrinogen antagonistic action and useful as an agent for the prevention and treatment of ischemic diseases such as thrombosis, cerebral infarction, myocardial infarction, etc...
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JPH0558608B2 |
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JPH0555489B2 |
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JPH05194333A |
PURPOSE: To industrially advantageously obtain ortho-amides by the reaction of alkoxymethylene iminium salts or formamidinium salts with alcoholates having a highly activated state. CONSTITUTION: Salts expressed by formula I are allowed ...
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JPH0530824B2 |
This invention relates to aryloxycycloalkanolaminoalkylene aryl ketones to the processes for their preparation and to their use as antihypertensive agents.
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JPH0578299A |
PURPOSE: To provide new compounds each of which has leukemia-inhibitory activity and shows a leukemia-inhibitory effect at the time of administrating it to a mammal suffered from leukemia and consists of 2,3,4,5- tetrahydroxybenzonitrile...
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JPH0516421B2 |
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JPH051780B2 |
Polyhydroxy-substituted benz, phenylacet and mandelamidines, amidates, amidoximes and hydroxyamidoximes-ribonucleotide reductase inhibitors, and free radical scavengers.
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JPH051784B2 |
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JPH05392B2 |
A process for preparing a compound of the formula : wherein R<2> is lower aliphatic hydrocarbon group which may be substituted with suitable substituent(s), cyclo(lower)alkyl or cyclo(lower)alkenyl; or a salt thereof, which comprises rea...
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JPH0479338B2 |
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JPH04352738A |
PURPOSE: To obtain an optically active chain terpenes which are useful intermediates in new production route for producing sarcophytol A having anticarcinogenic promoter action and antiulcer action at large quantity and at a low cost. CO...
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JPH04334351A |
PURPOSE: To obtain a biphenyl deriv. having useful pharmaceutical properties, especially an inhibiting effect on aggregation, and a pharmaceutical compsn. containing this compd. and to provide its preparation method. CONSTITUTION: The bi...
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JPH04326339A |
PURPOSE:To prevent deterioration due to moisture absorption or oxidization of an org. nonlinear optical material and to obtain a stable element as a laser light source against temp. or secular change by using at least one of a laser medi...
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JPH04305559A |
PURPOSE: To obtain a new compound having glycoprotein IIb/IIIa receptor antagonism, inhibitory action on blood platelet aggregation and antithrombotic action. CONSTITUTION: A compound shown by formula I (R1 is aryloxy (lower) alkanoyl; R...
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JPH04282356A |
PURPOSE: To readily produce the subject compound useful as an intermediate for various fine chemicals such as peptide antibiotics useful as drugs in a high yield, by subjecting an amidoxime derivative to an deoxidative reaction with CO i...
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JPH04273849A |
PURPOSE: To obtain a new fluorine-containing compound useful as a synthetic intermediate for agricultural chemicals and medicines or an active ingredient for agricultural chemicals and medicines. CONSTITUTION: A fluorine-containing compo...
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JPH04271139A |
PURPOSE: To improve the throughput of a single wafer semiconductor manufacturing equipment while restraining the equipment cost, which is equipped with the atmosphere side load lock chamber delivering wafers to a carrier cassette in the ...
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JPH0456821B2 |
Novel compounds of the formula which will be illustrated in greater detail in the description, their preparation and their use for controlling pests in crop protection are described.
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JPH04243855A |
PURPOSE: To provide the title new compound useful as an intermediate for fluorine-contg. amino acids, fluorine-contg. heterocyclic compounds, pesticides and drugs, also useful per se as a pesticide or men. CONSTITUTION: The objective com...
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JPH04221349A |
PURPOSE: To provide a new cyclophane which has the blood pressure lowering activity, coronary blood vessels dilating activity, and heartbeat rate lowering activity, and is effectively used in the therapy of hypertension and ischemic hear...
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JPH0439455B2 |
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JPH0459753A |
NEW MATERIAL:A compound of formula I (X, Y are H, halogen or lower alkyl). EXAMPLE: N-(α,α-Dimethyl-3-chloro)benzyl-N'-phenylamidine. USE: An antimicrobial agent for agriculture and horticulture. PREPARATION: An N-benzylformamide deriv...
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JPH03294255A |
NEW MATERIAL:A hydrazone compound shown by formula I [R1 is H, halogen, 1-4C alkyl and alkoxy, 1-4C haloalkyl, etc.; R2 is H, halogen or CH3 R3 is 1-4C alkyl; R4 is H, 1-6C alkenyl and haloalkyl; R5 is 1-6C alkyl and haloalkyl, 3-6C alke...
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JPH03264557A |
NEW MATERIAL:A compound expressed by formula I [R is substitutable phenyl, benzyl, alkoxycarbonyl or alkylcarbonyl; R1 is 2-10C alkyl, 1-6C alkyl having substituting group other than halogen, substitutable 2-6C alkenyl or alkinyl, hydraz...
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JPH03264565A |
NEW MATERIAL:A 5-[2'-(trans-4''-alkylcylcohexyl)ethyl]-2-(3,4-difluoropheny
l) pyrimidine shown by formula I (R is 1-10C straight-chain alkyl). EXAMPLE: 5-[2'-(trans-4''-Propylcylcohexyl)ethyl]-2-(3,4-difluorophen
yl)pyrimidine. USE: Use...
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JPH03503765A |
The invention is directed to azido-substituted octopamine agonists and the radiolabeled derivatives thereof. The invention also relates to past controlling compositions comprising the azido-substituted octopamine agonists of the inventio...
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JPH0354654B2 |
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JPH03169842A |
NEW MATERIAL:A compound of formula I [R1, R2 are alkyl; R3, R4 are H, CN, NO2, (halo)alkyl, cycloalkyl, (halo)alkoxy, (halo)alkylthio, alkylsulfonyl, alkylsulfinyl, phenyl, phenoxyalkyl, phenylthio, aminoalkyl, furfurylthio, amino, napht...
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JPH03135901A |
PURPOSE: To obtain a plant growth regulating agent containing amidinoformic acid derivative or salt thereof as active ingredient and inhibiting activity of phenylalanine ammonia lyase being rate-determining enzyme for biosynthesis of the...
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JPH03128350A |
NEW MATERIAL:A compound shown by formula I [(n) is 0-2; R3 is OH or dimethylamino; when R3 is OH and (n)=0, (i) R1 is methyl and R2 is 5- or 6-C, 4- or 5-F or 4-Br, (ii) R1 is F and R2 is 4-F, (iii) R1 is methoxy and R2 is 3-C, (iv) R1 i...
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JPH0310616B2 |
Amidine derivatives of the formula wherein R1 and R2, which may be the same or different, represent each a hydrogen atom or a lower alkyl group, or R1 and R2 together with an intermediary carbon atom and/or hetero atom may form a ring; X...
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JPH039902B2 |
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JPH037663B2 |
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JPH032856B2 |
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JPH02304066A |
PURPOSE: To obtain the title substance being an intermediate for the synthesis of pentafluoroethylpyrimidine economically by using a polyfloroalkylcarbonylacetic acid lower alkyl ester as a starting material and mixing and reacting this ...
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JPH0259145B2 |
Amidino compounds represented by the formula and pharmaceutically acceptable acid addition salts thereof are novel compounds and are useful as powerful antitrypsin, antiplasmin, antikallikrein and antithrombin agents. Having strong anti-...
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JPH0257062B2 |
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JPH0257061B2 |
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JPH0233031B2 |
The object of the present invention are new pharmacologically active substituted imidazolylphenyl amidines as H2 receptor blocking agents, which inhibit gastric acid secretion and which are useful antiulcer agents of the following formul...
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JPH0225902B2 |
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JPH02134398A |
NEW MATERIAL: A compd. (hydrate, isoster and salt) represented by formula I {wherein X is a group represented by formula II [wherein R4 is an α-amino acid residue; R5 is an α-amino acid residue or a peptide consisting of 2-4 α-amino a...
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JPH0219829B2 |
A method for preparing 6-amino-5-R3-2,4-diaminopyrimidine-3-oxides which comprises:
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JPH0216294B2 |
The invention relates to surface-active azo compounds obtainable by reacting azo compounds corresponding to the following general formula (I): (I) in which X and Y are the same or different and represent +TR and R represents C1-C4-alkyl,...
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JPH0291051A |
NEW MATERIAL: A compd. represented by formula I (wherein a wavy line means an E- or Z-isomer; R1 and R are each H, a protective group or combined together to form a protective group; R3 and R5 are each H, alkyl, alkenyl, cycloalkyl or ar...
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JPH0285244A |
NEW MATERIAL: Compd. of formula I (wherein A1 and A2 are each an acid, an ester, an amide, cyano or an aryl; and A3 is H, an alkyl, OH, a halogen, a nitro, an ether, A1 or A2) or their salts. EXAMPLE: N,N'-bis-(4-ethoxycarbonylphenyl)-2-...
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JPH0285241A |
PURPOSE: To provide a compd. used for preparing a medicine which has a specified compd. contg. a new compd. as an active ingredient and exhibits excellent bronchodilator activity and can be administered through various paths such as oral...
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JPH0285253A |
NEW MATERIAL: A compd. of formula I [wherein A is benzene which can have 1-4 substituents (which are 1-6C alkyl, 1-6C alkoxy, 1-6C alkenyloxy or the like), formula II, formula III or the like; X is O or NH; B is formula IV-formula VI; R ...
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JPH0276843A |
NEW MATERIAL: A compd. represented by formula I [wherein X1 to X6 are each CH or N; but at least one of X1 to X3 and X4 to X6 is CH; Y is NR5 (R5 is H or a lower alkyl), O or S; Z is NR6 (R6=R5), O or S; R2 and R4 are each R5 or R6; R1 a...
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