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JPH0254821B2 |
Tetrasubstituted urea and thiourea compounds useful as antiatherosclerotic agents, compositions thereof and processes for their preparation.
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JPH02256661A |
NEW MATERIAL: A benzoylthiourea compound represented by formula I, wherein A, B, X and Z represent F or Cl; (n) is 0 to 3; (p) is 0 or 1; Y is a haloalkyl; R1 represents H or SNR2R3, wherein R2 represents an alkyl; R3 represents an alkyl...
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JPH02235854A |
NEW MATERIAL:The compound of formula I (R1 is phenyl, naphthyl, thienyl or pyridyl; R2 is alkyl, alkoxyalkyl or cycloalkyl; R3 is H, alkyl, alkoxyalkyl, etc.; R4 is alkyl or cycloalkyl; Z is group of formula II, etc.; Y is group of formu...
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JPH0240064B2 |
The compounds of the formula I (I) in which R1 to R5 denote hydrogen; alkyl, alkoxy, alkylmercapto, alkylsulfinyl, alkylsulfonyl, alkylsulfonyloxy each of which can be halogenated, halogen or nitro, R6 to R10 denote hydrogen; alkyl, alko...
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JPH02221252A |
NEW MATERIAL: A compound represented by the formula I, wherein A, B denotes H or halogen, X denotes O or S, n is 0 to 4, Z denotes halogen or 1-6C alkyl, Y denotes 1-6C haloalkyl, 1-6C haloalkoxy, NO2, or CN, and Q denotes N or C-H, or, ...
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JPH02218642A |
NEW MATERIAL: A compd. represented by formula I (a group represented by formula II is divalent cyclic groups represented by formulae III-VII, R1 is 6- carboxyhexa-2-enyl or a modified group modified by the reduction of a double bond volu...
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JPH02193955A |
NEW MATERIAL: A compd. represented by formula (R1 is R7-CO-etc.; Z is amino acid; E is amino acid; Q is O or NR6; Y is -GtH2t-R13, etc.; R2, R5, R6 and R9 are each H or A; R3 and R13 are each H, A, Ar, etc.; R4 is (H or OH), etc.; R7 is ...
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JPH02188568A |
NEW MATERIAL: A compound given by formula I [(m) is 0, or 1; W is H, alkyl, alkenyl, alkynyl, or Ph(CH2)n-(Ph is phenyl; (n) is 0-2), R1NHCO-(R1 is H, or alkyl), R2CONH-(R2 is H, or alkyl); X is formula II ((p) is 0-2), -CONH-, =CSNH or ...
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JPH0231066B2 |
Substituted benzylcycloalkenylurea derivatives of the formula (I) (I) wherein X represents a halogen atom or a lower alkyl group, Y represents an oxygen atom or a sulfur atom, R1 represents a cycloalkenyl group and R2 represents a lower ...
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JPH0229074B2 |
Fungicidally active novel benzylurea derivatives of the formula in which R1 is a halogen atom or a lower alkyl group, X is an oxygen or sulfur atom, and R2 is an alkyl group, a cycloalkyl group having 5 to 8 carbon atoms, or a phenyl gro...
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JPH02152949A |
PURPOSE: To provide a compd. prohibiting protease encoded by HIV useful for preventing human immunedeficiency virus(HIV) infection and treating HIV infection and AIDS. CONSTITUTION: This HIV protease inhibitor is composed of a compd. rep...
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JPH02124868A |
PURPOSE: To obtain the compound useful as an intermediate for the synthesis of an antiulcerative famotidine in high yields by using a 3-substituted propionitrile and an oxonium salt as starting materials and reacting the product with a s...
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JPH0220639B2 |
The invention relates to compounds of the general formula (I) (I) and physiologically acceptable salts, N-oxides, hydrates and bioprecursors thereof, in which Y represents =O, =S, =CHNO2 or =NR3 where R3 represents hydrogen, nitro, cyano...
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JPH02117651A |
NEW MATERIAL:A compound of formula I (R1, R2 are alkyl, cycloalkyl; R3 through R6 are H, lower alkyl, cycloalkyl, aralkyl, pyridyl; X is O, S; n1, n2 are 1 to 6) or its salt. EXAMPLE: 1,3-Bis[[1-cycloheptyl-3-(2,4-difluorophenyl)ureido]m...
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JPH02115160A |
NEW MATERIAL: A compound of formula I (wherein R1 is H or a 1-4C alkyl; R2 is benzoyl, benzyl or α-hydroxybenzyl; R3 and R4 are each H, a 1-4C alkyl or an alkenyl or may be combined with the formamidine functional group to form a hetero...
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JPH0285247A |
NEW MATERIAL:An optically active 2-hydroxy-2-(substituted phenyl)ethylthiourea derivative expressed by formula I (R is lower alkyl). EXAMPLE: (+)-N-[2-Hydroxy-2-(chlorophenyl)ethyl]-N'-(methyl)thiourea.
USE: A medicine, having excellent...
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JPH0210823B2 |
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JPH0253774A |
NEW MATERIAL: A compound of formula I [wherein R1 is an alkyl, cycloalkyl, aryl, a heterocyclic ring; R2 is nitro, a halogen, alkyl, phenyl, etc.; R3 is alkyl, cyano and R3 can form a ring with R2; R4 is alkyl, alkenyl, phenyl, etc.; Y i...
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JPH026749B2 |
Novel N-aroyl N min -phenyl ureas having halogen or alkyl substituents in the 3- and 5-positions and haloalkyl, haloalkoxy or haloalkylthio in the 4-position of the N min -phenyl are more active and have a broader spectrum of effectivene...
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JPH025742B2 |
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JPH026469A |
NEW MATERIAL: A compound of formula I [wherein R1 is a (halogenated) 1-10C alkyl, a phenyl-1-7C alkyl or the like; R2 is a 1-10C alkyl, a 2-10C alkenyl, phenyl or the like; R3 is a 1-10C alkyl, alkoxy, a 3-7C cycloalkyl or the like; R4 i...
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JPH023666A |
NEW MATERIAL: A compound of formula I [wherein R1 is formula II or III; Z is O, CH2, NR8 or the like; E is a group composed of 0-2 amino acid molecules bonded through a peptide bond; Q is O or NR9; Y is CtH2t-R10, CtH2t- R11 or the like;...
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JPH024770A |
NEW MATERIAL: A compound represented by formula I [wherein R is an alkyl, a cycloalkyl or the like; A is formula II (wherein X is H, an alkyl, CF3, an alkoxyl or the like), formula III (wherein one of Y1 and Y2 is a halogen, methyl or ph...
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JPH024749A |
NEW MATERIAL: A compd. represented by formula I [wherein R1 are groups represented by formulae II, III, Z is Abu, Adu or Ala, E is a group having 0-2 amino acids bonded thereto by peptide formation, Q is 0 or NR, Y is CtH2t- R11 or CtH2t...
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JPH024703A |
PURPOSE: To use a specific compound as an active ingredient for controlling typical organisms of the order Acari such as mites, ticks and spider miles in animals and plants or on the animals and plants and insects. CONSTITUTION: A compou...
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JPH02141A |
NEW MATERIAL: An indan derivative of formula I [A is C=X (X is O, S); Y is N, N+-O--, CR8; R1, R2 are H, alkyl, or put together to be polymethylene; R3 is H, OH, alkoxy, acyloxy; R4 is H or put together with R3 to be single bond; when A ...
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JPH02250A |
NEW MATERIAL:A compound expressed by formula I {X1-X2 is -CH2-O-, etc.; L is -CH=CH or S; broken line is single bond or double bond; W is -S-, -O-, etc.; n is 0-3; Z is -NR1CO- (R1 is H, lower alkyl, etc.), etc.; Q is 1-18C alkyl, etc.; ...
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JPH021434A |
NEW MATERIAL: Compounds of formula I (R1 is formula II, formula III, NH-R2, etc.; R2 is H, amino, OC-Y, -P-phenyl-CH-Y, (substituted)alkyl, cycloalkyl, aryl, etc.; Y is EDTA, DTPA, DOTA, HETA, TRITA, TETA; M is a metal ion) or their salt...
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JPH02270A |
NEW MATERIAL: A compd. represented by formula I {wherein A is a group represented by formula II (wherein X is O or S) or groups represented by formula III, IV [wherein P5 is (halogenated) 1-5C alkyl], R1-R3 are H or halogen, R4 is haloge...
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JPH02703A |
PURPOSE: To obtain a treating agent containing one of specific compounds including new compounds as an active substance, exhibiting excellent stimulating effect on hematopoietic stem cells and capable of treating hematopoietic diseases s...
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JPH01311058A |
NEW MATERIAL:A compound shown by formula I [Q1 and Q2 are group shown by formula V (R1-R5 are H, halogen, trifluoromethyl, etc.) or group shown by formula VI; R6 and R7 are H, 1-6C alkyl, 1-6C alkenyl, 1-6C alkynyl, etc.; X is O or S]. E...
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JPH0154351B2 |
Complexes of pyromellitic diimide compounds which are ruminant feed additives and which improve feed efficiency are disclosed. The pyromellitic diimide compounds may be unsubstituted pyromellitic diimide itself, or one of the nitrogen at...
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JPH0153862B2 |
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JPH0153869B2 |
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JPH0149142B2 |
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JPH0148259B2 |
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JPH0147461B2 |
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JPH0144694B2 |
NEW MATERIAL:The titled compound of formula I (R1 is alkyl, cylohexyl or benzyl; R2 is alkyl, cyclohexyl or phenyl; R1 and R2 may together form a 5- membered, 6-membered or bicyclic hetero ring containing one N atom, two N atoms, or one ...
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JPH01233266A |
NEW MATERIAL:A benzoylurea derivative expressed by formula I (R is F or H; X is O or S then R is F and S when R is H). EXAMPLE: N-2,4,6-trifluorobenzoyl-N'-[2-fluoro-4-(1,1,2,2-tetrafluoro
ethoxy) phenyl]urea. USE: Useful as an insectici...
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JPH0140822B2 |
NEW MATERIAL:A compound of formulaI{Rf is 1-16C polyfluoroalkyl; A is trifunctional linking group; W is -Q2SO3M[Q2 is (CH2CH2)j (j is an integer 1-4), etc.; M is H, alkali metal, etc.], -Q2OSO3M, etc.; Q1 is (CH2) (l is an integer 2-6), ...
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JPH01168658A |
(57) [Abstract] Since this gazette is application data in front of an electronic application, the data of an abstract is not recorded.
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JPH01157944A |
NEW MATERIAL:The compound of formula I [X is group of formula II, III, etc.; R1WR4 are H, (substituted) alkyl or alkoxy, halogen, nitro, cyano, etc.; R5 and R6 are H, (substituted) alkyl or aryl, etc.; R7 is (substituted) alkyl, alkoxy, ...
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JPH01131148A |
NEW MATERIAL:A compound shown by formula I (R1 is Cl or F; R2 and R3 are F or H; at least one of R4, R5 and R6 is trifluoromethyl and the residue is Cl, F or H; X is O or S). EXAMPLE: N-2,6-Difluorobenzoyl-N'-3,5-dichloro-4-[3,5-(bistrif...
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JPH01131147A |
NEW MATERIAL:A compound shown by formula I (R1 is F or H; R2 is Cl or H; R3 is F, Br or lower haloalkyl; X and Y are O or S). EXAMPLE: N-2,6-Difluorobenzoyl-N'-3,5-dichloro-4-[4-(trifluoromethoxy
) anilino]phenylurea. USE: An insecticide...
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JPH0125740B2 |
The invention relates to new benzoylurea compounds of the general formula wherein R1 is a halogen atom, R2 is a hydrogen atom or a halogen atom, R3 is a hydrogen atom or represents 1 or 2 substituents which are selected from the group co...
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JPH0123459B2 |
Formamidine sulphides and disulphides endowed with herbicide activity are disclosed. The processes for their preparation, their use as herbicides and herbicidal compositions thereof are disclosed too.
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JPH0196164A |
NEW MATERIAL: A compd. of formula I (R1 is a (substd.) alkyl, an alkenyl, etc.; R2 is H, a (substd.) alkyl, etc.; R3 is H, a (substd.) alkyl, an alkinyl, etc.; X is O, S). EXAMPLE: N-Acetoamidemethyl-(E)-2-cyano-2-methoxyminoacetoamide. ...
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JPH0193569A |
NEW MATERIAL: A compd. of formula I [R1, R2 are each a 1 to 6C alkyl, F, Cl, Br, OR3 (R3 is a 1 to 6C alkyl, phenylmethyl); X is S, O; Y is O, NH; R4, R5 are each H, a 1 to 6C alkyl, or form a satd. carbon cyclic ring together with bonde...
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JPH0118895B2 |
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JPH0118896B2 |
A process for producing tolylthiourea having high purity comprises reacting toluidine with a thiocyanate and a mineral acid in the presence of an organic solvent and water.
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